SCHEMBL13806232

SCHEMBL13806232

Cn1cc(N)c2cccc(C(=O)O)c21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 1/20 0.44
CDC25B P30305 2/20 0.42
NR4A1 P22736 1/20 0.42
NR4A2 P43354 1/20 0.42
NR4A3 Q92570 1/20 0.42
FABP4 P15090 3/20 0.41
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
G6PD P11413 1/20 0.41
CASP7 P55210 1/20 0.41
CASP6 P55212 1/20 0.41
MYC P01106 2/20 0.39
DHODH Q02127 1/20 0.38
ALDH1A1 P00352 3/20 0.38
ALOX15 P16050 1/20 0.38
POLB P06746 1/20 0.37
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 2/20 0.37
NPC1 O15118 1/20 0.37
CASP3 P42574 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13806239 0.83 ALDH1A1 (0.56) NR4A2CASP7ALDH1A1KDM4EHSD17B10
SCHEMBL7868347 0.81 FABP4 (0.48) NR4A1NR4A2NR4A3FABP4S1PR1
SCHEMBL23809338 0.78 FABP4 (0.40) CDC25BNR4A1NR4A2NR4A3FABP4
SCHEMBL18975372 0.75 KDM4E (0.39) MMP2CDC25BCASP6ALDH1A1ALOX15
SCHEMBL70779 0.74 NR4A1 (0.50) CDC25BNR4A1NR4A2NR4A3FABP4
SCHEMBL13806534 0.73 MMP2 (0.44) MMP2NR4A2G6PDCASP7CASP6
SCHEMBL13806400 0.73 ALKBH5 (0.44) ALDH1A1ALOX15KDM4EHSD17B10NPC1
SCHEMBL13806312 0.72 BRD4 (0.40) ALDH1A1HSD17B10HPGD
SCHEMBL1094507 0.71 CDK2 (0.46) MYCALDH1A1POLBKDM4EHSD17B10
SCHEMBL7269233 0.70 PCSK9 (0.52) POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230330099-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2023-10-19 US disclosed
EP-2065382-A1 CGRP antagonists Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2009-06-03 EP disclosed
WO-2009050235-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed
WO-2009050237-A1 CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-04-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230330099-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL9 MMP2 3640/4885CDC25B 686/4885NR4A1 3610/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.