SCHEMBL1381409

SCHEMBL1381409

CC(C)c1nccc(NS(=O)(=O)N2CCCCC2)n1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
FKBP1A P62942 8/20 0.44
MAPK1 P28482 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
GLA P06280 1/20 0.41
KMT2A Q03164 1/20 0.41
PIK3C3 Q8NEB9 4/20 0.41
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
CXCR2 P25025 1/20 0.37
HRH4 Q9H3N8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23015779 0.76 CYP1A2 (0.40) MAPK1ALDH1A1LMNAHTTKMT2A
SCHEMBL5464187 0.71 FKBP1A (0.53) FKBP1AMAPK1ALDH1A1LMNAHTT
SCHEMBL5473695 0.71 FKBP1A (0.53) FKBP1AMAPK1ALDH1A1LMNAHTT
SCHEMBL30988530 0.70 PIK3C3 (0.46) FKBP1AMAPK1ALDH1A1LMNAHTT
SCHEMBL12356602 0.69 FLT3 (0.40) HRH4
SCHEMBL5476374 0.69 ALDH1A1 (0.46) FKBP1AMAPK1ALDH1A1LMNAHTT
SCHEMBL5473684 0.69 ALDH1A1 (0.46) FKBP1AMAPK1ALDH1A1LMNAHTT
SCHEMBL1380781 0.69 L3MBTL1 (0.55) ALDH1A1LMNAKMT2AKDM4E
SCHEMBL5474154 0.68 LMNA (0.58) FKBP1AMAPK1ALDH1A1LMNAHTT
SCHEMBL5471685 0.68 LMNA (0.58) FKBP1AMAPK1ALDH1A1LMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4809339-B2 2011-11-09 JP claimed
EP-1763517-B1 PYRIMIDINE DERIVATIVES AS 11BETA-HSD1 INHIBITORS HOFFMANN LA ROCHE (CH) 2011-05-11 EP claimed
EP-1763517-B1 PYRIMIDINE DERIVATIVES AS 11BETA-HSD1 INHIBITORS HOFFMANN LA ROCHE (CH) 2011-05-11 EP disclosed