SCHEMBL13845141

SCHEMBL13845141

Nc1cnc(CC[C@@H]2CCNC2)nc1NC1Cc2ccccc2C1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 3/20 0.34
PRKCQ Q04759 1/20 0.34
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
SLC6A3 Q01959 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13845148 0.94 HRH3 (0.38)
SCHEMBL13845160 0.76 KDM1A (0.41) GBA1PRKCQ
SCHEMBL13845192 0.76 PRKCQ (0.44) PRKCQ
SCHEMBL13845154 0.74 PRKCQ (0.46) GBA1PRKCQ
SCHEMBL21358959 0.65 HRH3 (0.42)
SCHEMBL13845246 0.64 TYRO3 (0.42) GBA1PRKCQ
SCHEMBL13845256 0.63 HRH4 (0.38) SLC6A2SLC6A4
SCHEMBL27987106 0.62 KDM1A (0.44) SLC6A2SLC6A4SLC6A3
SCHEMBL29290152 0.62 MAPK8 (0.43)
SCHEMBL3044569 0.61 GBA1 (0.56) GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009062059-A2 ISOMERIC PURINONES AND 1H-IMIDAZOPYRIDINONES AS PKC-THETA INHIBITORS PHARMACOPEIA, INC. (US) 2009-05-14 WO disclosed