SCHEMBL1385963

SCHEMBL1385963

CC(C)(C)c1ccc(S(=O)(=O)N2CCNC(C(=O)N(Cc3ccco3)C(=O)c3ccccc3)C2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.43
TSHR P16473 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
GAA P10253 3/20 0.40
LMNA P02545 2/20 0.40
HTT P42858 1/20 0.40
MAPT P10636 3/20 0.40
TP53 P04637 2/20 0.40
ALDH1A1 P00352 6/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
USP2 O75604 1/20 0.39
POLB P06746 3/20 0.38
TDP1 Q9NUW8 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
HPGD P15428 1/20 0.38
RECQL P46063 1/20 0.38
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041537 0.74 LMNA (0.53) KMT2AGAALMNATP53ALDH1A1
SCHEMBL4034634 0.70 ALDH1A1 (0.64) KMT2ATSHRNPSR1GAAMAPT
SCHEMBL4035135 0.67 POLB (0.42) KMT2ATSHRNPSR1GAALMNA
SCHEMBL26673580 0.63 ALDH1A1 (0.49) KMT2ALMNAALDH1A1SMN1; SMN2HPGD
SCHEMBL13997348 0.62 LMNA (0.48) KMT2ATSHRGAALMNAHTT
SCHEMBL735124 0.62 LMNA (0.66) KMT2AGAALMNAHTTTP53
SCHEMBL6267145 0.61 SMN1; SMN2 (0.60) KMT2ATSHRLMNAHTTMAPT
SCHEMBL27780939 0.61 ALDH1A1 (0.50) KMT2ALMNAHTTALDH1A1POLB
SCHEMBL22501790 0.61 TRPV4 (0.60) KMT2ATSHRLMNAMAPTTP53
SCHEMBL8288240 0.61 DPP4 (0.55) TSHRLMNAHTTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4825664-B2 2011-11-30 JP claimed
EP-1592389-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES Applied Research Systems ARS Holding N.V. (AN) 2005-11-09 EP claimed
WO-2004071390-A2 PIPERAZINE-2-CARBOXAMIDE DERIVATIVES APPLIED RESEARCH SYSTEMS ARS HOLDING N.V. (AN) 2004-08-26 WO claimed