SCHEMBL13860906

SCHEMBL13860906

CCCCNc1ccc(-c2nnc(-c3ncccn3)nn2)nc1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TYRO3 Q06418 11/20 0.41
MERTK Q12866 11/20 0.41
FLT3 P36888 10/20 0.41
GAS6 Q14393 10/20 0.41
AXL P30530 4/20 0.41
RRM2 P31350 1/20 0.40
TLR8 Q9NR97 3/20 0.39
TLR7 Q9NYK1 2/20 0.39
NPC1 O15118 1/20 0.37
HCAR3 P49019 1/20 0.36
KCNH3 Q9ULD8 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
KCNH2 Q12809 1/20 0.35
UTS2R Q9UKP6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12468718 0.86 MERTK (0.44) TYRO3MERTKFLT3GAS6AXL
SCHEMBL21553939 0.76 SMN1; SMN2 (0.49)
SCHEMBL23636379 0.75 RAB9A (0.39) NPC1
SCHEMBL13736761 0.75 RAB9A (0.54) NPC1
SCHEMBL25912779 0.74 TRPM8 (0.41) CYP3A4CYP2D6KCNH2
SCHEMBL13830642 0.72 RAB9A (0.37) NPC1
SCHEMBL19010907 0.71 NPC1 (0.46) NPC1CYP3A4CYP2D6
SCHEMBL29401898 0.71 HIF1A (0.42)
SCHEMBL14197601 0.71 RRM2 (0.48) RRM2TLR8TLR7NPC1HCAR3
SCHEMBL15748102 0.70 HPGDS (0.48) NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2709668-A1 BIO-ORTHOGONAL DRUG ACTIVATION Koninklijke Philips N.V. (NL) 2014-03-26 EP disclosed
WO-2012156920-A1 BIO-ORTHOGONAL DRUG ACTIVATION KONINKLIJKE PHILIPS ELECTRONICS N.V. (NL) 2012-11-22 WO disclosed