SCHEMBL13875868

SCHEMBL13875868

COc1ccc(-n2c(=O)[nH]c3c(N4CCNCC4)nc(Cl)nc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 10/20 0.48
ALDH1A1 P00352 10/20 0.48
CASP1 P29466 8/20 0.48
CASP7 P55210 8/20 0.48
HSD17B10 Q99714 3/20 0.48
CYP2C9 P11712 1/20 0.48
USP2 O75604 8/20 0.47
CYP3A4 P08684 5/20 0.47
HTR3E A5X5Y0 1/20 0.47
HTR3B O95264 1/20 0.47
ADRB1 P08588 1/20 0.47
HTR3A P46098 1/20 0.47
HTR3D Q70Z44 1/20 0.47
HTR3C Q8WXA8 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
HIF1A Q16665 7/20 0.46
TP53 P04637 3/20 0.46
LMNA P02545 2/20 0.46
MAPK1 P28482 4/20 0.46
HPGD P15428 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13875865 0.85 SLC2A1 (0.45) CYP1A2ALDH1A1CASP1CASP7HSD17B10
SCHEMBL13876126 0.84 CSNK2A1 (0.41) CYP1A2ALDH1A1CASP1CASP7HSD17B10
SCHEMBL13875754 0.81 HTR2C (0.39) CYP1A2CYP2C9CYP3A4HTR3EHTR3B
SCHEMBL13876137 0.80 CYP1A2 (0.36) CYP1A2ALDH1A1HSD17B10CYP2C9USP2
SCHEMBL13875756 0.79 CHRNB2 (0.45) CYP1A2ALDH1A1CYP2C9CYP3A4HTR3E
SCHEMBL13875683 0.78 SLC2A1 (0.53) CYP1A2ALDH1A1CASP1CASP7HSD17B10
SCHEMBL13875885 0.76 SLC2A1 (0.42) CYP1A2ALDH1A1CASP1CASP7HSD17B10
SCHEMBL13866874 0.75 DPP4 (0.42) CYP1A2ALDH1A1CASP1CASP7HSD17B10
SCHEMBL13866907 0.74 CYP1A2 (0.42) CYP1A2ALDH1A1CASP1CASP7HSD17B10
SCHEMBL13876148 0.72 CHRNB2 (0.43) CYP1A2ALDH1A1CASP1CASP7HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7524847-B2 Fused 1,3-dihydro-imidazole ring compounds EISAI R&D MANAGEMENT CO., LTD. (JP) 2009-04-28 US disclosed