SCHEMBL1388928

SCHEMBL1388928

Fc1ccc2occ(CN3CCC=C(C=Cc4ccccc4)C3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.39
ALDH1A1 P00352 4/20 0.36
HSD17B10 Q99714 1/20 0.36
DRD2 P14416 2/20 0.36
DRD3 P35462 2/20 0.36
RAB9A P51151 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
TSHR P16473 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
MAPK1 P28482 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
KDM1A O60341 1/20 0.33
HTR6 P50406 1/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8858347 0.84 HTR1A (0.47) HTR1ADRD2DRD3SMN1; SMN2KDM4E
SCHEMBL8858346 0.84 HTR1A (0.47) HTR1ADRD2DRD3SMN1; SMN2KDM4E
SCHEMBL1388879 0.73 DRD2 (0.44) HTR1AALDH1A1HSD17B10DRD2DRD3
SCHEMBL11805239 0.72 SIGMAR1 (0.47) ALDH1A1DRD2RAB9ASIGMAR1KDM4E
SCHEMBL11805236 0.72 SIGMAR1 (0.47) ALDH1A1DRD2RAB9ASIGMAR1KDM4E
SCHEMBL8791055 0.71 MAOA (0.45) HTR1ADRD2DRD3RAB9ASIGMAR1
SCHEMBL8858349 0.71 MAOA (0.45) HTR1ADRD2DRD3RAB9ASIGMAR1
SCHEMBL8858342 0.70 DRD2 (0.48) HTR1ADRD2DRD3RAB9ASIGMAR1
SCHEMBL8858344 0.70 DRD2 (0.48) HTR1ADRD2DRD3RAB9ASIGMAR1
SCHEMBL11793066 0.68 SIGMAR1 (0.40) ALDH1A1RAB9ASIGMAR1MAPK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-H09512542-A 1997-12-16 JP claimed
EP-0757686-A1 BENZOFURAN DERIVATIVES AS D 4? RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LTD. (GB) 1997-02-12 EP claimed
WO-1995029911-A1 BENZOFURAN DERIVATIVES AS D4 RECEPTOR ANTAGONISTS MERCK SHARP & DOHME LIMITED (GB) 1995-11-09 WO claimed