SCHEMBL13891716

SCHEMBL13891716

COc1ccccc1CN1CCCOc2nc(SC)nc(-c3ccccc3C)c2C1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 3/20 0.37
MAOB P27338 1/20 0.37
GAA P10253 3/20 0.37
KDM4E B2RXH2 2/20 0.37
RECQL P46063 1/20 0.37
TACR1 P25103 2/20 0.35
USP2 O75604 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ACHE P22303 1/20 0.35
MAPT P10636 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALDH1A1 P00352 2/20 0.35
TSHR P16473 2/20 0.35
POLB P06746 1/20 0.35
HTR7 P34969 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13891714 0.88 ADORA2A (0.40) ADORA2AMAOBGAAKDM4ERECQL
SCHEMBL13891686 0.86 MAPT (0.35) MAPTMEN1KMT2ATSHRCYP3A4
SCHEMBL13891740 0.71 TLR7 (0.36) MEN1KMT2ATSHRCYP3A4CYP2C19
SCHEMBL13891713 0.68 TACR1 (0.42) TACR1
SCHEMBL13891767 0.68 P2RX3 (0.40) ACHEMEN1KMT2AALDH1A1NPSR1
SCHEMBL13891721 0.67 HTT (0.37) GAAKDM4EMAPTMEN1KMT2A
SCHEMBL13891766 0.65 KDM4E (0.38) KDM4ETACR1HSD17B10MAPTMEN1
SCHEMBL5236630 0.65 TACR1 (0.37) KDM4ETACR1MAPTALDH1A1
SCHEMBL13891688 0.64 TACR1 (0.41) TACR1KMT2ATSHR
SCHEMBL5230109 0.63 TACR1 (0.39) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1473295-B1 FUSED BICYCLIC PYRIMIDINE DERIVATIVES KYORIN SEIYAKU KK (JP) 2009-04-01 EP disclosed