SCHEMBL14025577

SCHEMBL14025577

CCN(CC)CCOc1ccc(CN(C)S(=O)(=O)c2cccc(CNCc3ccccc3)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
CYP1A2 P05177 1/20 0.50
LTA4H P09960 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
BCHE P06276 6/20 0.45
ACHE P22303 6/20 0.45
TAS2R14 Q9NYV8 1/20 0.44
MAOB P27338 1/20 0.42
MMP1 P03956 2/20 0.42
MMP9 P14780 2/20 0.42
MMP13 P45452 2/20 0.42
MEN1 O00255 1/20 0.42
MAPT P10636 1/20 0.42
KMT2A Q03164 1/20 0.42
KCNH2 Q12809 1/20 0.42
MCHR1 Q99705 1/20 0.42
ALDH1A1 P00352 1/20 0.41
HCRTR2 O43614 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14025558 0.90 TDP1 (0.44) HTTCYP1A2LTA4HCYP2D6CYP2C9
SCHEMBL14025581 0.85 RAB9A (0.53) HTTCYP1A2LTA4HCYP2D6CYP2C9
SCHEMBL14025560 0.83 ALDH1A1 (0.53) HTTTAS2R14MEN1MAPTKMT2A
SCHEMBL14025582 0.79 HRH3 (0.49) HTTCYP1A2LTA4HCYP2D6CYP2C9
SCHEMBL14025600 0.77 ALDH1A1 (0.50) HTTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14025559 0.77 ALDH1A1 (0.50) HTTCYP1A2LTA4HCYP2D6CYP2C9
SCHEMBL14025614 0.76 ALDH1A1 (0.53) HTTCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL14025570 0.75 CASP3 (0.49) HTTTAS2R14MEN1KMT2AALDH1A1
SCHEMBL14068043 0.75 MEN1 (0.44) HTTTAS2R14MEN1MAPTKMT2A
SCHEMBL14025548 0.74 PKM (0.53) HTTMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea METASTATIX, INC. 2008-10-23 US disclosed
WO-2008109154-A1 CHEMOKINE RECEPTOR MODULATORS ALTIRIS THERAPEUTICS, INC. (US) 2008-09-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080261978-A1 treating or preventing HIV infections, and in treating proliferative disorders such as inhibiting the metastasis of various cancers; 1-(4-((pyridin-2-ylmethylamino)methyl)benzyl)-3-phenylurea MKI67, CCNI, CDKN1A HTT 4443/4885CYP1A2 1066/4885LTA4H 3640/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.