SCHEMBL14096743

SCHEMBL14096743

COC(=O)C(NC(=O)[C@@H](NC(=O)OCc1ccccc1)C1CCCCC1)C(C)(C)C

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
CYP3A4 P08684 2/20 0.47
TSHR P16473 2/20 0.47
MAPT P10636 1/20 0.47
TP53 P04637 1/20 0.47
CTSK P43235 3/20 0.46
CTSL P07711 1/20 0.46
CTSB P07858 1/20 0.46
CTSS P25774 1/20 0.46
MMP2 P08253 2/20 0.45
EPHX1 P07099 1/20 0.45
MBOAT4 Q96T53 1/20 0.45
MMP3 P08254 1/20 0.45
ALOX15 P16050 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
CYP1A2 P05177 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL464127 1.00 ALDH1A1 (0.47) ALDH1A1CYP3A4TSHRMAPTTP53
SCHEMBL464269 0.93 ALDH1A1 (0.47) ALDH1A1CYP3A4TSHRMAPTTP53
SCHEMBL13201867 0.88 ALDH1A1 (0.48) ALDH1A1CYP3A4TSHRMAPTTP53
SCHEMBL15087458 0.87 CTSK (0.48) ALDH1A1CYP3A4TSHRMAPTTP53
SCHEMBL20825664 0.85 EPHX1 (0.56) ALDH1A1CYP3A4TSHRMAPTTP53
SCHEMBL13219417 0.85 MEN1 (0.47) ALDH1A1CYP3A4TSHRMAPTCTSK
SCHEMBL8372704 0.84 CTSB (0.61) CTSKCTSLCTSBCTSS
SCHEMBL13219700 0.84 CTSK (0.44) ALDH1A1CYP3A4TSHRMAPTTP53
SCHEMBL8667196 0.82 TRPM8 (0.54) ALDH1A1CTSKCTSLCTSBCTSS
SCHEMBL20681662 0.81 CTSL (0.54) ALDH1A1CYP3A4TSHRCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1958956-A2 Peptidomimetic protease inhibitors Vertex Pharmaceuticals Incorporated (US) 2008-08-20 EP disclosed