SCHEMBL14102007

SCHEMBL14102007

Cc1cc(-c2cnco2)cc(-c2nn(-c3cc(NCCC(=O)O)ccc3S(C)(=O)=O)c(=O)c3ncccc23)c1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
IMPDH2 P12268 2/20 0.33
NAMPT P43490 2/20 0.32
PTK2 Q05397 1/20 0.31
NTRK1 P04629 1/20 0.31
CCR9 P51686 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4721114 0.93 NAMPT (0.31) IMPDH2NAMPTPTK2NTRK1
SCHEMBL4721371 0.93 PTK2 (0.33) IMPDH2NAMPTPTK2CCR9
SCHEMBL4721609 0.89 PTK2 (0.33) IMPDH2NAMPTPTK2CCR9
SCHEMBL4722289 0.88 IMPDH2 (0.36) IMPDH2NAMPTPTK2CCR9
SCHEMBL4719259 0.83 L3MBTL1 (0.33) IMPDH2CCR9
SCHEMBL4720352 0.82 NAMPT (0.30) NAMPT
SCHEMBL4724113 0.82 MAPT (0.37) IMPDH2NAMPTPTK2
SCHEMBL4720084 0.81 NAMPT (0.33) IMPDH2NAMPTPTK2NTRK1
SCHEMBL4722805 0.80 MAPT (0.40) NAMPT
SCHEMBL4720681 0.80 JAK2 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed