SCHEMBL4720084

SCHEMBL4720084

Cc1cc(-c2cnco2)cc(-c2nn(-c3cc(NCCO)ccc3C(F)(F)F)c(=O)c3ncccc23)c1

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.33
TRPV1 Q8NER1 1/20 0.32
S1PR1 P21453 2/20 0.32
S1PR3 Q99500 2/20 0.32
NTRK1 P04629 1/20 0.31
PTK2 Q05397 1/20 0.31
IMPDH2 P12268 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
IMPDH1 P20839 1/20 0.31
TACR1 P25103 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
SCD O00767 1/20 0.30
QPCT Q16769 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4722805 0.88 MAPT (0.40) NAMPTALDH1A1LMNAPOLBMAPT
SCHEMBL4723141 0.86 MAPT (0.39) NAMPTPTK2IMPDH2ALDH1A1LMNA
SCHEMBL4722197 0.86 MEN1 (0.32) TRPV1TACR1
SCHEMBL4719909 0.86 TRPV1 (0.35) TRPV1ALDH1A1LMNAPOLBTACR1
SCHEMBL4723705 0.82 TRPV1 (0.30) TRPV1
SCHEMBL4721659 0.81 RIOK2 (0.35)
SCHEMBL4723349 0.81 PTK2 (0.30) PTK2
SCHEMBL4724221 0.81 NTRK1 (0.33) NTRK1PTK2IMPDH2IMPDH1QPCT
SCHEMBL14102007 0.81 IMPDH2 (0.33) NAMPTNTRK1PTK2IMPDH2
SCHEMBL4722896 0.80 TRPV1 (0.32) TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed
EP-1953147-A1 HETEROCYCLIC COMPOUND AND MEDICINAL APPLICATION THEREOF Japan Tobacco, Inc. (JP) 2008-08-06 EP disclosed