SCHEMBL14148384

SCHEMBL14148384

NC(=O)Nc1sc(-c2ccccc2)nc1-c1ccccc1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.73
ALDH1A1 P00352 3/20 0.73
MAPT P10636 3/20 0.73
POLB P06746 2/20 0.56
GAA P10253 1/20 0.56
NTRK1 P04629 2/20 0.54
CDC7 O00311 4/20 0.54
DBF4 Q9UBU7 4/20 0.54
CCNE1 P24864 1/20 0.54
CDK2 P24941 1/20 0.54
PTGDR2 Q9Y5Y4 3/20 0.51
KMT2A Q03164 2/20 0.51
NPSR1 Q6W5P4 1/20 0.51
IKBKB O14920 1/20 0.49
JAK2 O60674 1/20 0.49
JAK3 P52333 1/20 0.49
RARA P10276 1/20 0.48
RARB P10826 1/20 0.48
RARG P13631 1/20 0.48
TBK1 Q9UHD2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27519692 0.92 KDM4E (0.67) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL4268936 0.87 KDM4E (0.77) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL4738310 0.83 ALDH1A1 (0.71) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL5556366 0.83 TBK1 (0.55) KDM4EALDH1A1MAPTGAAIKBKB
SCHEMBL11652002 0.82 MAPT (0.69) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL14148528 0.81 KDM4E (0.68) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL4737628 0.79 KDM4E (0.64) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL14148405 0.77 ALDH1A1 (0.67) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL4737640 0.77 KDM4E (0.63) KDM4EALDH1A1MAPTPOLBGAA
SCHEMBL14148414 0.77 ALDH1A1 (0.63) KDM4EALDH1A1MAPTNTRK1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008090382-A1 THIAZOLE AND OXAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PRION DISEASES, CANCER AND CONDITIONS OF THE CENTRAL NERVOUS SYSTEM AS WELL AS IN THE REGULATION OF STEM CELLS THE UNIVERSITY OF SHEFFIELD (GB) 2008-07-31 WO disclosed