SCHEMBL1414841

SCHEMBL1414841

CN1Cc2c(ccc3cc(C(C)(O)c4cn(C(c5ccccc5)(c5ccccc5)c5ccccc5)cn4)ccc23)C1=O

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 5/20 0.49
CYP2C8 P10632 1/20 0.49
CYP3A4 P08684 2/20 0.33
CASR P41180 1/20 0.30
UGCG Q16739 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1414881 0.89 CYP17A1 (0.45) CYP17A1CYP2C8CYP3A4
SCHEMBL1414812 0.89 CYP17A1 (0.58) CYP17A1CYP2C8CYP3A4
SCHEMBL1414934 0.80 CYP17A1 (0.41) CYP17A1CYP2C8
SCHEMBL1414829 0.79 CYP17A1 (0.58) CYP17A1CYP2C8CYP3A4
SCHEMBL5751159 0.73 ACSS2 (0.39) CYP17A1CASR
SCHEMBL1415054 0.73 CYP17A1 (0.57) CYP17A1CYP2C8CYP3A4
SCHEMBL8540731 0.72 KIF11 (0.46) CYP3A4
SCHEMBL4025339 0.71 CYP17A1 (0.53) CYP17A1CYP3A4CASR
SCHEMBL31285478 0.70 ENPP2 (0.36)
SCHEMBL1414930 0.70 CYP17A1 (0.70) CYP17A1CYP2C8CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1344777-B1 IMIDAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE TAKEDA PHARMACEUTICAL (JP) 2011-03-16 EP disclosed
US-6960586-B2 Imidazole derivatives, process for their preparation and their use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2005-11-01 US disclosed
US-20040024039-A1 Imidazole derivatives, process for their preparation and their use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2004-02-05 US disclosed
EP-1344777-A1 IMIDAZOLE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE Takeda Chemical Industries, Ltd. (JP) 2003-09-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040024039-A1 Imidazole derivatives, process for their preparation and their use CYP17A1, HSD17B7, CYP51A1 CYP17A1 1/4885CYP2C8 137/4885CYP3A4 203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.