SCHEMBL14158201

SCHEMBL14158201

CC(C)C[C@H](NC(=O)/C=C/c1ccccc1)C(=O)Cn1nc(CCc2ccccc2)oc1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C9 P11712 2/20 0.47
CYP1A2 P05177 1/20 0.47
MAPK1 P28482 1/20 0.47
CYP2C19 P33261 1/20 0.47
CASP1 P29466 1/20 0.45
CASP3 P42574 1/20 0.45
CASP7 P55210 1/20 0.45
CASP6 P55212 1/20 0.45
CASP8 Q14790 1/20 0.45
GAA P10253 2/20 0.41
LMNA P02545 2/20 0.41
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
RECQL P46063 2/20 0.40
NOS2 P35228 6/20 0.40
NOS3 P29474 4/20 0.40
NOS1 P29475 4/20 0.40
TAS1R3 Q7RTX0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4868592 0.84 CTSK (0.43) LMNAHTTSMN1; SMN2TAS1R3TAS1R1
SCHEMBL4869837 0.79 CTSL (0.44) ALDH1A1CYP2C9CYP1A2CYP2C19SMN1; SMN2
SCHEMBL4868064 0.78 CTSK (0.47) ALDH1A1CASP1CASP3CASP7CASP6
SCHEMBL4869933 0.78 KMT2A (0.41) ALDH1A1SMN1; SMN2MMP1POLBMMP2
SCHEMBL4866588 0.78 CTSS (0.48) CASP1CASP3CASP7CASP6CASP8
SCHEMBL14158062 0.75 KMT2A (0.51) ALDH1A1CYP3A4CYP2C9CYP1A2MAPK1
SCHEMBL5493122 0.75 CASP1 (0.48) ALDH1A1CYP3A4CYP2C9CYP1A2MAPK1
SCHEMBL14597548 0.75 CASP1 (0.48) ALDH1A1CYP3A4CYP2C9CYP1A2MAPK1
SCHEMBL4868071 0.74 CASP3 (0.38) CASP3
SCHEMBL4912638 0.72 MEN1 (0.52) ALDH1A1CASP1CASP3CASP7CASP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7390804-B2 N-containing five-membered ring compounds and pharmaceutical agents comprising the same as active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-06-24 US disclosed
US-7390804-B2 N-containing five-membered ring compounds and pharmaceutical agents comprising the same as active ingredient ONO PHARMACEUTICAL CO., LTD. (JP) 2008-06-24 US disclosed