SCHEMBL14166129

SCHEMBL14166129

O=C(OCc1ccccc1)c1cc(O)cc(Br)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.62
TDP1 Q9NUW8 3/20 0.62
SLC6A2 P23975 1/20 0.62
SLC6A3 Q01959 1/20 0.62
LMNA P02545 3/20 0.61
RAB9A P51151 5/20 0.55
NPC1 O15118 3/20 0.55
TSHR P16473 1/20 0.51
ALDH1A1 P00352 4/20 0.50
MAPT P10636 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
HPGD P15428 2/20 0.50
GAA P10253 1/20 0.49
CA12 O43570 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
CA14 Q9ULX7 1/20 0.49
MEN1 O00255 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9166162 0.89 TDP1 (0.72) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL9696689 0.89 TDP1 (0.72) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL5094893 0.88 KMT2A (0.62) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL20078314 0.85 KMT2A (0.58) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL26007966 0.85 KMT2A (0.58) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL5094821 0.85 KMT2A (0.58) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL26736622 0.85 KMT2A (0.58) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL5101575 0.85 KMT2A (0.58) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL21924208 0.84 KMT2A (0.66) KMT2ATDP1SLC6A2SLC6A3LMNA
SCHEMBL20472063 0.84 KMT2A (0.59) KMT2ATDP1SLC6A2SLC6A3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 49 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12458706-B2 Compounds and therapeutic uses thereof AVVINITY THERAPEUTICS LIMITED (GB) 2025-11-04 US disclosed
CN-113382771-B Compounds and therapeutic uses thereof 阿维尼蒂治疗有限公司 2025-01-24 CN disclosed
CN-110753558-B Novel compounds and therapeutic uses thereof 森陶里治疗有限公司 2023-10-24 CN disclosed
US-11766483-B2 Compounds and therapeutics uses thereof Centauri Therapeutics Limited (GB/GB) (GB) 2023-09-26 US disclosed
US-11766483-B2 Compounds and therapeutics uses thereof Centauri Therapeutics Limited (GB/GB) (GB) 2023-09-26 US disclosed
US-11766483-B2 Compounds and therapeutics uses thereof Centauri Therapeutics Limited (GB/GB) (GB) 2023-09-26 US disclosed
EP-3606561-B1 NOVEL COMPOUNDS AND THERAPEUTIC USES THEREOF CENTAURI THERAPEUTICS LTD (GB) 2023-08-02 EP disclosed
EP-3606561-B1 NOVEL COMPOUNDS AND THERAPEUTIC USES THEREOF CENTAURI THERAPEUTICS LTD (GB) 2023-08-02 EP disclosed
CN-108472381-B Compounds and therapeutic uses thereof 森陶里治疗有限公司 2023-06-06 CN disclosed
US-20220162262-A1 NOVEL COMPOUNDS AND THERAPEUTIC USES THEREOF Centauri Therapeutics Limited (GB/GB) (GB) 2022-05-26 US disclosed
EP-2718280-B1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY CHIESI FARMA SPA (IT) 2015-09-16 EP disclosed
EP-2718280-B1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY CHIESI FARMA SPA (IT) 2015-09-16 EP disclosed
US-8877774-B2 Compounds having muscarinic receptor antagonist and beta2 Adrenergic receptor agonist activity CHIESI FARMACEUTICI S.P.A. (IT) 2014-11-04 US disclosed
US-8877774-B2 Compounds having muscarinic receptor antagonist and beta2 Adrenergic receptor agonist activity CHIESI FARMACEUTICI S.P.A. (IT) 2014-11-04 US disclosed
US-8877774-B2 Compounds having muscarinic receptor antagonist and beta2 Adrenergic receptor agonist activity CHIESI FARMACEUTICI S.P.A. (IT) 2014-11-04 US disclosed
EP-2718280-A1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY Chiesi Farmaceutici S.p.A. (IT) 2014-04-16 EP disclosed
US-20130045169-A1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY CHIESI FARMACEUTICI S.P.A. (IT) 2013-02-21 US disclosed
US-20130045169-A1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY CHIESI FARMACEUTICI S.P.A. (IT) 2013-02-21 US disclosed
WO-2012168359-A1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY CHIESI FARMACEUTICI S.P.A. (IT) 2012-12-13 WO disclosed
WO-2012168359-A1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY CHIESI FARMACEUTICI S.P.A. (IT) 2012-12-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12458706-B2 Compounds and therapeutic uses thereof MAVS, NFATC1, MYD88 KMT2A 3895/4885TDP1 2967/4885SLC6A2 4811/4885
US-20130045169-A1 COMPOUNDS HAVING MUSCARINIC RECEPTOR ANTAGONIST AND BETA2 ADRENERGIC RECEPTOR AGONIST ACTIVITY ADRB2, ADRB1, ADRA2B KMT2A 3123/4885TDP1 4410/4885SLC6A2 1397/4885
US-11766483-B2 Compounds and therapeutics uses thereof MAVS, MYD88, CD47 KMT2A 3577/4885TDP1 2480/4885SLC6A2 4830/4885
US-20220162262-A1 NOVEL COMPOUNDS AND THERAPEUTIC USES THEREOF MAVS, MYD88, CD47 KMT2A 4285/4885TDP1 2941/4885SLC6A2 4757/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.