SCHEMBL14200465

SCHEMBL14200465

CCC(CC)N(C(=O)CC(C)(C)C)c1cccc(C)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
ALDH1A1 P00352 4/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
PAX8 Q06710 2/20 0.41
TP53 P04637 1/20 0.41
GPX4 P36969 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 3/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
JAK2 O60674 1/20 0.40
HSD17B1 P14061 3/20 0.40
HSD17B2 P37059 3/20 0.40
POLQ O75417 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14200479 0.89 TAS1R3 (0.44) HPGDMEN1KMT2AALDH1A1RAB9A
SCHEMBL14200504 0.89 KMT2A (0.43) HPGDMEN1KMT2AALDH1A1RAB9A
SCHEMBL14200771 0.87 HTT (0.35) HPGDMEN1KMT2AHTTNPSR1
SCHEMBL14200503 0.87 ALDH1A1 (0.46) HPGDMEN1KMT2AALDH1A1RAB9A
SCHEMBL14200440 0.84 ALDH1A1 (0.44) HPGDALDH1A1RAB9ANPC1CYP2C19
SCHEMBL14200452 0.84 SIGMAR1 (0.37) ALDH1A1TDP1SMN1; SMN2HDAC8HDAC6
SCHEMBL14200818 0.84 RIPK1 (0.42) HPGDMEN1KMT2AALDH1A1RAB9A
SCHEMBL14200458 0.84 TAS1R3 (0.42) HPGDMEN1KMT2AALDH1A1RAB9A
SCHEMBL14200460 0.83 MTNR1B (0.36) KMT2AHDAC6
SCHEMBL14200493 0.83 LTB4R2 (0.40) MEN1KMT2AALDH1A1TP53CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed