SCHEMBL14200537

SCHEMBL14200537

O=c1[nH]cc(CC2CCc3c(Cl)cccc32)[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
HTR2C P28335 1/20 0.35
MAPT P10636 2/20 0.34
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
DAO P14920 1/20 0.33
NOTUM Q6P988 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HTT P42858 1/20 0.31
ALOX5 P09917 1/20 0.31
FFAR1 O14842 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31
OPRK1 P41145 1/20 0.31
OPRL1 P41146 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
CMA1 P23946 1/20 0.30
DRD2 P14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1337944 0.85 ADRA2A (0.40) ESR1ESR2ALDH1A1FFAR1OPRM1
SCHEMBL1340047 0.85 ESR1 (0.36) ESR1ESR2HTR2C
SCHEMBL1339435 0.79 HTR6 (0.48)
SCHEMBL29107353 0.75 HRH4 (0.42)
SCHEMBL1340184 0.74 ESR1 (0.57) ESR1ESR2MAPTOPRM1
SCHEMBL1339428 0.74 ADRA2A (0.40) OPRM1
SCHEMBL1337725 0.72 SRD5A1 (0.39) ESR1ESR2ALDH1A1
SCHEMBL1339442 0.72 SRD5A1 (0.39) ESR1ESR2ALDH1A1
SCHEMBL1340622 0.72 SRD5A1 (0.39) ESR1ESR2ALDH1A1
SCHEMBL1339993 0.72 SRD5A1 (0.39) ESR1ESR2FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080091028-A1 IMIDAZOLE-2-THIONES ALLERGAN, INC. (US) 2008-04-17 US disclosed
US-20080091028-A1 IMIDAZOLE-2-THIONES ALLERGAN, INC. (US) 2008-04-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080091028-A1 IMIDAZOLE-2-THIONES ADRB2, ADRA2C, ADRA2B ESR1 1836/4885ESR2 180/4885HTR2C 119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.