SCHEMBL14218480

SCHEMBL14218480

CC(=O)Nc1cccc2c(C(=O)N3CC4(C)CC(C)(C)CC34)c[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.40
PGR P06401 1/20 0.40
NR3C2 P08235 1/20 0.40
AR P10275 1/20 0.40
AVPR1A P37288 7/20 0.38
ERCC1 P07992 1/20 0.37
FEN1 P39748 1/20 0.37
ERCC4 Q92889 1/20 0.37
PARP14 Q460N5 2/20 0.37
CNR2 P34972 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
BRPF1 P55201 1/20 0.34
AVPR2 P30518 2/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
NR4A2 P43354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13668476 0.74 NR3C1 (0.40) NR3C1PGRNR3C2ARAVPR1A
SCHEMBL14218514 0.73 NR4A2 (0.45) AVPR1ACNR2NPSR1NR4A2
SCHEMBL14218550 0.72 CNR2 (0.45) AVPR1ACNR2AVPR2
SCHEMBL14218479 0.71 NR4A2 (0.50) NPSR1ALDH1A1KMT2ANR4A2
SCHEMBL14218551 0.70 MEN1 (0.45) CNR2ALDH1A1KMT2A
SCHEMBL14218512 0.69 HTR3E (0.35) AVPR1ACNR2NPSR1AVPR2ALDH1A1
SCHEMBL14218513 0.67 HPGD (0.45) ALDH1A1KMT2A
SCHEMBL11982194 0.65 CYP2C9 (0.50) ALDH1A1KMT2A
SCHEMBL10267219 0.64 CYP2C19 (0.69)
SCHEMBL3456247 0.62 AVPR2 (0.63) AVPR1ANPSR1AVPR2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080108598-A1 Pharmaceutical use of substituted amides NOVO NORDISK A/S (DK) 2008-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080108598-A1 Pharmaceutical use of substituted amides HSD11B1, HSD3B1, HSD11B2 NR3C1 33/4885PGR 985/4885NR3C2 40/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.