SCHEMBL14229202

SCHEMBL14229202

CCCCN(CCOC)S(=O)(=O)CC(F)(F)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.34
CES1 P23141 4/20 0.33
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
PKM P14618 1/20 0.32
CYP2C19 P33261 1/20 0.32
MLYCD O95822 1/20 0.31
CACNA1B Q00975 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14228926 0.89 CES1 (0.40) CES1MLYCD
SCHEMBL14228929 0.85 CA1 (0.39) CES1MLYCD
SCHEMBL14230124 0.82 CES1 (0.34) RORCCES1
SCHEMBL14200414 0.82 CNR1 (0.32) RORC
SCHEMBL14200216 0.80 CES1 (0.34) CES1
SCHEMBL14229348 0.79 BMP1 (0.32) CES1CYP1A2CYP3A4CYP2C9PKM
SCHEMBL14229197 0.78 CES1 (0.35) CES1MLYCD
SCHEMBL14229149 0.77 BMP1 (0.41) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL14229686 0.76 PIK3CD (0.35) CYP1A2CYP3A4CYP2C9PKMCYP2C19
SCHEMBL14229525 0.76 CNR2 (0.38) CYP1A2CYP3A4CYP2C9PKMCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7365093-B2 Endothelin antagonists ABBOTT LABORATORIES (US) 2008-04-29 US disclosed
US-7208517-B1 Endothelin antagonists ABBOTT LABORTORIES (US) 2007-04-24 US disclosed