SCHEMBL14237644

SCHEMBL14237644

COc1ccccc1-c1ccc2cccc(-n3ccnc3C)c2n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41
P2RX4 Q99571 1/20 0.40
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
PDE10A Q9Y233 2/20 0.38
KCNN4 O15554 1/20 0.38
CYP19A1 P11511 1/20 0.38
HSP90AA1 P07900 1/20 0.37
STK10 O94804 1/20 0.37
SLK Q9H2G2 1/20 0.37
BDKRB2 P30411 1/20 0.37
ALDH1A1 P00352 2/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2036823 0.77 MCHR1 (0.57) MAOAMAOBPDE10ACYP19A1HSP90AA1
SCHEMBL10904420 0.77 GAA (0.47) ALDH1A1LMNACYP3A4TSHRMEN1
SCHEMBL728248 0.76 MAOA (0.64) MAOAMAOBP2RX4CYP11B1CYP11B2
SCHEMBL1672334 0.76 PDE10A (0.57) MAOAMAOBPDE10ACYP19A1HSP90AA1
Hydrochloric Acid SCHEMBL1901179 0.75 MAOA (0.63) MAOAMAOBP2RX4CYP11B1CYP11B2
SCHEMBL3192555 0.75 ALDH1A1 (0.52) MAOAMAOBCYP19A1HSP90AA1ALDH1A1
Hydrochloric Acid SCHEMBL28789582 0.74 PDE10A (0.56) MAOAMAOBPDE10ACYP19A1HSP90AA1
Hydrochloric Acid SCHEMBL2953393 0.74 PDE10A (0.56) MAOAMAOBPDE10ACYP19A1HSP90AA1
SCHEMBL38654702 0.72 AR (0.49) MAOAMAOBPDE10AKCNN4HSP90AA1
SCHEMBL9731132 0.70 KCNN4 (0.47) P2RX4KCNN4ALDH1A1LMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2315588-B1 6-1H-IMIDAZO-QUINAZOLINE AND QUINOLINES DERIVATIVES, NEW MAO INHIBITORS AND IMIDAZOLINE RECEPTOR LIGANDS ROTTAPHARM SPA (IT) 2012-12-19 EP claimed