SCHEMBL14246766

SCHEMBL14246766

O=C(Nc1sc2ccccc2c1Cl)NC1CCCc2ccccc21

nearest known ligand 0.60

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 3/20 0.60
TAS1R1 Q7RTX1 3/20 0.60
LMNA P02545 2/20 0.60
KMT2A Q03164 4/20 0.59
MEN1 O00255 1/20 0.59
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 1/20 0.58
GAA P10253 1/20 0.58
HPGD P15428 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
PRSS12 P56730 2/20 0.56
NPSR1 Q6W5P4 1/20 0.55
EPHX1 P07099 1/20 0.53
TAS1R2 Q8TE23 1/20 0.51
CNR1 P21554 1/20 0.51
CNR2 P34972 1/20 0.51
HTT P42858 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14246768 0.82 PRSS12 (0.70) TAS1R3TAS1R1LMNAKMT2AALDH1A1
SCHEMBL701314 0.76 TAS1R3 (1.00) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL11748653 0.72 KMT2A (0.67) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL11746591 0.72 KMT2A (0.70) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL11746602 0.72 KMT2A (0.70) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL24334864 0.71 HTT (0.68) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL15824830 0.71 HTT (0.68) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL703637 0.71 TAS1R3 (1.00) TAS1R3TAS1R1LMNAKMT2AMEN1
Hydrochloric Acid SCHEMBL11745237 0.71 KMT2A (0.68) TAS1R3TAS1R1LMNAKMT2AMEN1
SCHEMBL11271580 0.70 KMT2A (0.64) TAS1R3TAS1R1LMNAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9334256-B2 Agents and methods for treating ischemic and other diseases NONO INC. (CA) 2016-05-10 US disclosed
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases NONO INC. (CA) 2014-08-07 US disclosed
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases NONO INC. (CA) 2014-08-07 US disclosed
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases NONO INC. (CA) 2014-08-07 US disclosed
EP-2720695-A2 AGENTS AND METHODS FOR TREATING ISCHEMIC AND OTHER DISEASES NoNO Inc. (CA) 2014-04-23 EP disclosed
WO-2012174488-A2 AGENTS AND METHODS FOR TREATING ISCHEMIC AND OTHER DISEASES NONO, INC. (CA) 2012-12-20 WO disclosed
WO-2012174488-A2 AGENTS AND METHODS FOR TREATING ISCHEMIC AND OTHER DISEASES NONO, INC. (CA) 2012-12-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221423-A1 Agents And Methods For Treating Ischemic And Other Diseases TRPM7, TRPM8, TRPM5 TAS1R3 2049/4885TAS1R1 2229/4885LMNA 2548/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.