SCHEMBL1426328

SCHEMBL1426328

O=C(c1cccc(CO)c1)c1ccc(F)c(F)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
VNN1 O95497 3/20 0.47
PRSS1 P07477 1/20 0.46
PRSS2 P07478 1/20 0.46
PRSS3 P35030 1/20 0.46
CNR2 P34972 1/20 0.46
KMT2A Q03164 1/20 0.44
SMYD3 Q9H7B4 1/20 0.43
ACHE P22303 1/20 0.43
HSD17B14 Q9BPX1 2/20 0.41
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27982785 0.86 PRSS1 (0.59) PRSS1PRSS2PRSS3CNR2SMYD3
SCHEMBL1002846 0.84 CES2 (0.53) CES2CES1VNN1KMT2AACHE
SCHEMBL7046114 0.80 L3MBTL1 (0.65) PRSS1PRSS2PRSS3CNR2SMYD3
SCHEMBL7967901 0.80 CES2 (0.73) CES2CES1VNN1KMT2AHSD17B14
SCHEMBL4710159 0.79 MAOB (0.44) CES2CES1VNN1KMT2A
SCHEMBL13664920 0.79 CES2 (0.47) CES2CES1VNN1ACHEHSD17B14
SCHEMBL332679 0.78 ATM (0.61) CES2CES1VNN1KMT2AACHE
SCHEMBL14409543 0.77 VNN1 (0.55) VNN1PRSS1PRSS2PRSS3CNR2
SCHEMBL13664921 0.77 CES2 (0.53) CES2CES1VNN1KMT2AHSD17B14
SCHEMBL5937441 0.77 CYP11B1 (0.57) CES1CNR2KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2301936-A1 SPIRODIAMINE-DIARYLKETOXIME DERIVATIVE Banyu Pharmaceutical Co., Ltd. (JP) 2011-03-30 EP disclosed
US-20110071129-A1 SPIRODIAMINE-DIARYL KETOXIME DERIVATIVE MSD K.K. (JP) 2011-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110071129-A1 SPIRODIAMINE-DIARYL KETOXIME DERIVATIVE MCHR2, MCHR1, ADRB2 CES2 2405/4885CES1 1844/4885VNN1 3228/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.