SCHEMBL1428237

SCHEMBL1428237

C1CCN(N2CCC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.38
ALDH1A1 P00352 2/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
CA1 P00915 3/20 0.32
CA2 P00918 3/20 0.32
HRH3 Q9Y5N1 1/20 0.32
POLB P06746 1/20 0.32
F2 P00734 1/20 0.30
CA12 O43570 1/20 0.30
CA9 Q16790 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL285244 1.00 MGLL (0.38) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL13836035 1.00 MGLL (0.38) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL2457046 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL513824 0.95
SCHEMBL2807354 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL3658220 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL42220 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL726729 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL6926105 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1
SCHEMBL14084740 0.95 MGLL (0.40) MGLLALDH1A1TSHRKMT2ACA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 78 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025124516-A1 COMPOUND HAVING AKT KINASE-DEGRADING ACTIVITY, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL USE THEREOF 南京正大天晴制药有限公司 2025-06-19 WO claimed
CN-120157686-A Compound with AKT kinase degradation activity, preparation method and pharmaceutical application thereof 南京正大天晴制药有限公司 2025-06-17 CN claimed
WO-2024012570-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL USE THEREOF 西藏海思科制药有限公司 2024-01-18 WO claimed
CN-117229263-A Compound for inhibiting or degrading Bcl6 and application of compound in medicine 四川海思科制药有限公司 2023-12-15 CN claimed
WO-2023232133-A1 COMPOUND FOR INHIBITING OR DEGRADING BCL6 AND USE THEREOF IN PHARMACEUTICS 西藏海思科制药有限公司 2023-12-07 WO claimed
WO-2023208165-A1 NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL APPLICATION THEREOF 四川海思科制药有限公司 2023-11-02 WO claimed
CN-116947877-A Benzimidazole derivative and application thereof in medicine 四川海思科制药有限公司 2023-10-27 CN claimed
CN-111372931-B Heterocyclic compounds as protein kinase inhibitors 怡诺安有限公司 2023-03-24 CN claimed
WO-2023016518-A1 HETEROCYCLIC DERIVATIVE, AND COMPOSITION AND PHARMACEUTICAL USE THEREOF 四川海思科制药有限公司 2023-02-16 WO claimed
CN-114874286-A Compound for degrading BTK kinase, pharmaceutical composition and pharmaceutical application thereof 四川海思科制药有限公司 2022-08-09 CN claimed
WO-2008006032-A1 CYCLOPENTA [D] PYRIMIDINES AS AKT PROTEIN KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2008-01-10 WO claimed
EP-1707563-A2 Methods and compositions utilizing quinazolinones Cytokinetics, Inc. (US) 2006-10-04 EP claimed
EP-1686120-A2 Methods and compositions utilizing quinazolinones Cytokinetics, Inc. (US) 2006-08-02 EP claimed
US-20040023996-A1 Methods and compositions utilizing quinazolinones CYTOKINETICS, INC. 2004-02-05 US claimed
US-6562831-B1 Inhibitors of the mitotic kinesin KSP and are useful in the treatment of cellular proliferative diseases CYTOKINETICS, INC. 2003-05-13 US claimed
EP-1296959-A1 METHODS AND COMPOSITIONS UTILIZING QUINAZOLINONES Cytokinetics, Inc. (US) 2003-04-02 EP claimed
WO-2001030768-A9 METHODS AND COMPOSITIONS UTILIZING QUINAZOLINONES CYTOKINETICS INC (US) 2002-08-15 WO claimed
EP-1226129-A1 METHODS AND COMPOSITIONS UTILIZING QUINAZOLINONES Cytokinetics, Inc. (US) 2002-07-31 EP claimed
WO-2001098278-A1 METHODS AND COMPOSITIONS UTILIZING QUINAZOLINONES CYTOKINETICS, INC. (US) 2001-12-27 WO claimed
WO-2001030768-A1 METHODS AND COMPOSITIONS UTILIZING QUINAZOLINONES CYTOKINETICS, INC. (US) 2001-05-03 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040023996-A1 Methods and compositions utilizing quinazolinones KIF5B, KIF5C, KIF2C MGLL 4578/4885ALDH1A1 1628/4885TSHR 4831/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.