SCHEMBL14286147

SCHEMBL14286147

O=C(c1cc(-n2nnnc2-c2ccc(F)c(F)c2F)c[nH]1)N1CCCC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.37
MAPK10 P53779 1/20 0.37
GRIN2B Q13224 5/20 0.36
ALPL P05186 4/20 0.35
ALDH1A1 P00352 4/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 3/20 0.35
CYP3A4 P08684 2/20 0.35
HPGD P15428 2/20 0.35
CYP2D6 P10635 2/20 0.35
KMT2A Q03164 2/20 0.35
MEN1 O00255 1/20 0.35
CYP1A2 P05177 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
LMNA P02545 2/20 0.33
KDM4E B2RXH2 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5042176 0.81 ALDH1A1 (0.39) ALDH1A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL10067969 0.80 HRH4 (0.35) GRIN2BALDH1A1CYP2C9CYP2C19HPGD
SCHEMBL14286149 0.78 MAPK1 (0.41) MAPK1MAPK10ALPLALDH1A1HPGD
SCHEMBL14286161 0.71 ALDH1A1 (0.36) ALDH1A1CYP2C9CYP2C19CYP3A4CYP2D6
SCHEMBL14600770 0.68 HRH4 (0.36) ALDH1A1HPGDF2F10LMNA
SCHEMBL5038382 0.63 MAPK1 (0.49) MAPK1MAPK10GRIN2BALPLALDH1A1
SCHEMBL14286171 0.63 MAPK1 (0.52) MAPK1MAPK10GRIN2BALPLALDH1A1
SCHEMBL986040 0.63 KCNN4 (0.40) MAPK1ALDH1A1HPGDKMT2AMEN1
SCHEMBL14286136 0.63 MAPK1 (0.44) MAPK1MAPK10GRIN2BALDH1A1HPGD
SCHEMBL14286148 0.63 MAPK1 (0.42) MAPK1MAPK10ALDH1A1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed