SCHEMBL14286152

SCHEMBL14286152

O=C1N=NC(c2c[nH]c(C(=O)Nc3ncc[nH]3)c2)=C1c1cccc(F)c1F

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK7 Q13164 12/20 0.37
MAPK14 Q16539 6/20 0.37
RPS6KA3 P51812 2/20 0.34
DYRK1A Q13627 2/20 0.34
DCLK1 O15075 1/20 0.34
DYRK3 O43781 1/20 0.34
ROCK2 O75116 1/20 0.34
PRKD3 O94806 1/20 0.34
MAP4K4 O95819 1/20 0.34
ABL1 P00519 1/20 0.34
EGFR P00533 1/20 0.34
NTRK1 P04629 1/20 0.34
LCK P06239 1/20 0.34
FYN P06241 1/20 0.34
CDK1 P06493 1/20 0.34
CSF1R P07333 1/20 0.34
LYN P07948 1/20 0.34
SRC P12931 1/20 0.34
MARK3 P27448 1/20 0.34
AXL P30530 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600769 0.82 CCNE2 (0.34) RPS6KA3PTGESCCNE2CCNE1CDK2
SCHEMBL14286161 0.73 ALDH1A1 (0.36) MAPK7MAPK14PTGESYTHDC1
SCHEMBL14286160 0.68 CHRM1 (0.42) ROCK2GSK3BROCK1
SCHEMBL14286157 0.66 MAPK1 (0.56) GSK3B
SCHEMBL10067972 0.64 KCNN4 (0.34) RPS6KA3DYRK1ADCLK1DYRK3ROCK2
SCHEMBL14286146 0.64 ADRA2A (0.37) MAPK7MAPK14PTGESCDK2CCNC
SCHEMBL6825870 0.62 NPC1 (0.54)
SCHEMBL1126571 0.61 FGFR3 (0.42) PTGES
SCHEMBL14310378 0.61 PTGES (0.37) MAPK7PTGESCDK2
SCHEMBL5038382 0.59 MAPK1 (0.49) DYRK1AWNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed