SCHEMBL14286155

SCHEMBL14286155

O=C(NCC1CCCO1)c1cc(-n2nnnc2-c2ccccc2F)c[nH]1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
ALDH1A1 P00352 6/20 0.51
HPGD P15428 6/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2C19 P33261 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.48
KDM4E B2RXH2 1/20 0.48
HSD17B10 Q99714 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
LMNA P02545 1/20 0.46
MAPK1 P28482 1/20 0.45
MAPK10 P53779 1/20 0.45
GSK3B P49841 1/20 0.45
KCNH2 Q12809 1/20 0.45
HTT P42858 2/20 0.45
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10067973 0.83 RAB9A (0.51) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL14278771 0.80 MAPK1 (0.49) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL5037115 0.79 GSK3B (0.51) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL5037119 0.79 GSK3B (0.51) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL14286176 0.77 HPGD (0.52) ALDH1A1HPGDCYP1A2CYP2C19L3MBTL1
SCHEMBL14286150 0.75 GSK3B (0.51) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL14286159 0.74 ALDH1A1 (0.41) NPC1RAB9AALDH1A1MEN1KMT2A
SCHEMBL10067975 0.72 ALDH1A1 (0.46) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL14286127 0.71 GSK3B (0.56) NPC1RAB9AALDH1A1HPGDCYP1A2
SCHEMBL14278769 0.71 GSK3B (0.55) NPC1RAB9AALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed
US-7314885-B2 Pyrrole compounds useful as kinase inhibitors VERTEX PHARMACEUTICALS INCORPORATED (US) 2008-01-01 US disclosed