Medrylamine

Medrylamine

SCHEMBL142910

COc1ccc(C(OCCN(C)C)c2ccccc2)cc1

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.78
SLC6A4 P31645 6/20 0.78
SLC6A3 Q01959 6/20 0.78
LMNA P02545 4/20 0.78
CHRM2 P08172 4/20 0.78
CYP2D6 P10635 4/20 0.78
ADRA2A P08913 3/20 0.78
CHRM1 P11229 3/20 0.78
OPRM1 P35372 3/20 0.78
DRD3 P35462 3/20 0.78
ADRA2B P18089 3/20 0.78
HRH1 P35367 3/20 0.78
KCNH2 Q12809 3/20 0.78
CHRM4 P08173 2/20 0.78
CHRM5 P08912 2/20 0.78
CHRM3 P20309 2/20 0.78
HRH2 P25021 2/20 0.78
HTR2A P28223 2/20 0.78
HTR2C P28335 2/20 0.78
ADRA1A P35348 2/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenhydramine SCHEMBL12543374 0.88 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL4064 0.88 SLC6A2 (1.00) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL11795332 0.87 SLC6A2 (0.96) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL29205078 0.87 SLC6A2 (0.96) SLC6A2SLC6A4SLC6A3LMNACHRM2
SCHEMBL4670285 0.87 SCN1A (0.55) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL25219551 0.87 SLC6A2 (0.96) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL10487818 0.87 LMNA (1.00) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL9565209 0.87 SLC6A2 (0.96) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL17071 0.87 LMNA (1.00) SLC6A2SLC6A4SLC6A3LMNACHRM2
Diphenhydramine SCHEMBL28210970 0.87 SLC6A2 (0.96) SLC6A2SLC6A4SLC6A3LMNACHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 298 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8026285-B2 Control release of biologically active compounds from multi-armed oligomers BEZWADA BIOMEDICAL, LLC (US) 2011-09-27 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
US-20090076174-A1 CONTROL RELEASE OF BIOLOGICALLY ACTIVE COMPOUNDS FROM MULTI-ARMED OLIGOMERS BEZWADA BIOMEDICAL, LLC (US) 2009-03-19 US claimed
CN-101330905-A Freeze-drying process and products obtained thereby SCIDOSE LLC (US) 2008-12-24 CN claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
EP-1829527-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-09-05 EP claimed
EP-1829528-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-09-05 EP claimed
EP-1815846-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-08-08 EP claimed
EP-1815847-A2 Aggregate with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2007-08-08 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
US-20050282879-A1 Methods and composition for treatment of migraine and symptoms thereof SALEHANI FOAD 2005-12-22 US claimed
EP-1551370-A1 AGGREGATE WITH INCREASED DEFORMABILITY, COMPRISING AT LEAST THREE AMPHIPATS, FOR IMPROVED TRANSPORT THROUGH SEMI-PERMEABLE BARRIERS AND FOR THE NON-INVASIVE DRUG APPLICATION IN VIVO, ESPECIALLY THROUGH THE SKIN IDEA AG (DE) 2005-07-13 EP claimed
US-20040105881-A1 Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin IDEA AG (DE) 2004-06-03 US claimed
WO-2004032900-A1 AGGREGATE WITH INCREASED DEFORMABILITY, COMPRISING AT LEAST THREE AMPHIPATS, FOR IMPROVED TRANSPORT THROUGH SEMI-PERMEABLE BARRIERS AND FOR THE NON-INVASIVE DRUG APPLICATION IN VIVO, ESPECIALLY THROUGH THE SKIN IDEA AG (DE) 2004-04-22 WO claimed
EP-1336602-A1 Nitrate prodrugs able to release nitric oxide in a controlled and selective way and their use for prevention and treatment of inflammatory, ischemic and proliferative diseases Scaramuzzino, Giovanni (IT) 2003-08-20 EP claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050282879-A1 Methods and composition for treatment of migraine and symptoms thereof HRH3, HRH4, HNMT SLC6A2 641/4885SLC6A4 558/4885SLC6A3 1630/4885
US-20090076174-A1 CONTROL RELEASE OF BIOLOGICALLY ACTIVE COMPOUNDS FROM MULTI-ARMED OLIGOMERS MME, CTSA, ALG1 SLC6A2 4524/4885SLC6A4 4418/4885SLC6A3 4221/4885
US-20040105881-A1 Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin CUTA, ABCG2, PIGS SLC6A2 98/4885SLC6A4 264/4885SLC6A3 195/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.