SCHEMBL14334591

SCHEMBL14334591

NC(=O)c1cccnc1OCCN1CCCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.50
DRD1 P21728 1/20 0.50
DRD3 P35462 1/20 0.50
PARP1 P09874 2/20 0.49
DHODH Q02127 1/20 0.49
LTA4H P09960 4/20 0.49
CHRNB2 P17787 1/20 0.49
CHRNA4 P43681 1/20 0.49
RAB9A P51151 1/20 0.47
BCHE P06276 4/20 0.46
ACHE P22303 2/20 0.46
MEN1 O00255 1/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
PSMB1 P20618 1/20 0.46
PSMB5 P28074 1/20 0.46
PSMB2 P49721 1/20 0.46
ABCB1 P08183 1/20 0.45
PTGS2 P35354 1/20 0.45
GCGR P47871 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4708251 0.88 GAA (0.50) PARP1MEN1GAAKMT2A
SCHEMBL14334593 0.80 CHRNB2 (0.54) LTA4HCHRNB2CHRNA4PTGS2
SCHEMBL876068 0.79 DRD2 (0.69) DRD2DRD1DRD3MEN1GAA
SCHEMBL15477409 0.79 CYP2C19 (0.46) PARP1DHODH
SCHEMBL14377256 0.79 LTA4H (0.50) DRD2DRD1DRD3LTA4HCHRNB2
SCHEMBL6302948 0.77 RAB9A (0.55) PARP1RAB9A
SCHEMBL3729269 0.76 ALDH1A1 (0.55) PARP1RAB9AMEN1KMT2A
SCHEMBL6304815 0.76 RAB9A (0.54) PARP1RAB9AMEN1KMT2A
SCHEMBL29786652 0.76 ALDH1A1 (0.55) PARP1RAB9AMEN1KMT2A
SCHEMBL17979955 0.76 ALDH1A1 (0.59) DRD2DRD1DRD3PARP1DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012176123-A1 3 - IMIDAZOLYL- INDOLES FOR THE TREATMENT OF PROLIFERATIVE DISEASES NOVARTIS AG (CH) 2012-12-27 WO disclosed