SCHEMBL14404661

SCHEMBL14404661

CCCCOc1ccc2c(c1)CCN(c1ccc(F)cc1)C2Cc1ccc(C)c([N+](=O)[O-])c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA9 Q16790 2/20 0.37
CA14 Q9ULX7 2/20 0.37
CA7 P43166 1/20 0.37
PPARA Q07869 5/20 0.36
PPARG P37231 2/20 0.36
PPARD Q03181 3/20 0.35
HTR1A P08908 1/20 0.35
HTR1D P28221 1/20 0.35
HTR1B P28222 1/20 0.35
MCHR1 Q99705 1/20 0.35
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
DRD2 P14416 2/20 0.35
HTR6 P50406 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14382001 0.89 ESR1 (0.43) ESR1ESR2
SCHEMBL14404649 0.88 SIGMAR1 (0.41) CA1CA2CA9CA14CA7
SCHEMBL14404660 0.85 PPARA (0.36) PPARAPPARGPPARDS1PR1S1PR3
SCHEMBL14051060 0.81 ESR1 (0.42) PPARAPPARGPPARDMCHR1ESR1
SCHEMBL14404651 0.81 ESR1 (0.42) CA1CA2CA9CA14CA7
SCHEMBL14051122 0.81 ESR1 (0.41) PPARAPPARDESR1ESR2DRD2
SCHEMBL14404749 0.78 CYP3A4 (0.43) PPARAPPARGPPARDMCHR1ESR1
SCHEMBL14382000 0.76 MMP1 (0.41) ESR1ESR2
SCHEMBL14404514 0.76 MEN1 (0.39) PPARAPPARGPPARDESR1ESR2
SCHEMBL14404513 0.76 BCHE (0.42) PPARAPPARGPPARDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279489-B2 Compounds and methods for modulation of estrogen receptors SIGNAL PHARMACEUTICALS, LLC (US) 2007-10-09 US disclosed