SCHEMBL14415965

SCHEMBL14415965

O=C1c2ncccc2CCc2cccc(Cl)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 2/20 0.41
CDC25B P30305 2/20 0.41
MAPK14 Q16539 1/20 0.40
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NSD2 O96028 3/20 0.39
THRB P10828 2/20 0.39
BLM P54132 2/20 0.39
TDP2 O95551 1/20 0.39
ABL1 P00519 1/20 0.39
PLCG1 P19174 1/20 0.39
CES1 P23141 1/20 0.39
PAX8 Q06710 1/20 0.39
RIN1 Q13671 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
GAA P10253 1/20 0.39
PTAFR P25105 2/20 0.38
FNTA P49354 4/20 0.38
FNTB P49356 4/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002677 0.76 LMNA (0.43) S100A4CDC25BNSD2LMNASMN1; SMN2
SCHEMBL7255792 0.73 CES1 (0.61) MAPK14MEN1KMT2ANSD2THRB
SCHEMBL4095527 0.72 HRH1 (0.49) S100A4CDC25BMAPK14MEN1KMT2A
SCHEMBL29413038 0.72 HRH1 (0.60) MAPK14MEN1KMT2APTAFRFNTA
SCHEMBL4968772 0.72 CDC25B (0.41) CDC25BKMT2ABLMCES1KDM4E
SCHEMBL3839936 0.72 HRH1 (0.60) MAPK14MEN1KMT2APTAFRFNTA
SCHEMBL2456241 0.71 TDP2 (0.45) S100A4CDC25BMAPK14MEN1KMT2A
SCHEMBL29439737 0.71 TDP2 (0.45) S100A4CDC25BMAPK14MEN1KMT2A
SCHEMBL568118 0.71 AHR (0.41) CES1ABCB1ADRA2AADRA2BADRA2C
SCHEMBL8118609 0.69 MAOA (0.46) S100A4CDC25BMAPK14MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070213340-A1 Farnesyl protein transferase inhibitors SCHERING CORPORATION 2007-09-13 US disclosed
US-20070213340-A1 Farnesyl protein transferase inhibitors SCHERING CORPORATION 2007-09-13 US disclosed
WO-2007084498-A1 PIPERAZINE DERIVATIVES AS FARNESYL PROTEIN TRANSFERASE INHIBITORS SCHERING CORPORATION (US) 2007-07-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213340-A1 Farnesyl protein transferase inhibitors FNTB, FNTA, FDPS S100A4 1090/4885CDC25B 793/4885MAPK14 1655/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.