SCHEMBL1442844

SCHEMBL1442844

N#Cc1cccc(C(F)(F)F)n1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSS P25774 4/20 0.51
IRAK4 Q9NWZ3 2/20 0.48
P2RX7 Q99572 1/20 0.40
SOS2 Q07890 1/20 0.39
NOTUM Q6P988 1/20 0.39
CTSK P43235 2/20 0.38
SYK P43405 2/20 0.38
IDH1 O75874 2/20 0.38
TGFBR1 P36897 1/20 0.38
IDH2 P48735 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30449276 1.00 CTSS (0.51) CTSSIRAK4P2RX7SOS2NOTUM
SCHEMBL17200145 0.85 IRAK4 (0.43) CTSSIRAK4P2RX7CTSKSYK
SCHEMBL24794162 0.84 CTSS (0.49) CTSSIRAK4SOS2CTSKIDH1
SCHEMBL2960222 0.79 CTSK (0.41) CTSSIRAK4SOS2CTSKIDH1
SCHEMBL2514328 0.79 P2RX7 (0.43) CTSSIRAK4P2RX7NOTUMIDH1
SCHEMBL30627137 0.79 P2RX7 (0.40) CTSSIRAK4P2RX7NOTUMIDH1
SCHEMBL19873380 0.79 P2RX7 (0.40) CTSSIRAK4P2RX7NOTUMIDH1
SCHEMBL25305047 0.78 CTSS (0.41) CTSSIRAK4P2RX7SOS2CTSK
SCHEMBL995983 0.77 SOS2 (0.50) CTSSSOS2CTSKIDH1
SCHEMBL3295150 0.77 P2RX7 (0.50) P2RX7NOTUMIDH1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 106 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103874685-B Process for the preparation of 4-amino-3-chloro-5-fluoro-6- (substituted) pyridine-2-carboxylic acid esters DOW AGROSCIENCES LLC (US) 2016-02-03 CN claimed
CN-103458689-B The preparation method of 4-amino-5-fluorine-3-halo-6-(replacement) pyridine-2-manthanoate DOW AGROSCIENCES LLC (US) 2015-09-23 CN claimed
CN-103429082-B Process for the preparation of 4-amino-3-chloro-5-fluoro-6-(substituted)picolinates DOW AGROSCIENCES LLC 2015-05-06 CN claimed
CN-103458689-A Process for the preparation of 4-amino-5-fluoro-3-halo-6-(substituted)picolinates DOW AGROSCIENCES LLC 2013-12-18 CN claimed
CN-103429082-A Process for the preparation of 4-amino-3-chloro-5-fluoro-6-(substituted)picolinates DOW AGROSCIENCES LLC 2013-12-04 CN claimed
US-12433895-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2025-10-07 US disclosed
US-20240335448-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE PHARMARESROUCES (SHANGHAI) CO., LTD. (CN) 2024-10-10 US disclosed
WO-2024126619-A1 ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING A COMPOUND OF FORMULA (I) AND A COMPOUND OF FORMULA (II), AND DISPLAY DEVICE COMPRISING THE ORGANIC ELECTROLUMINESCENT DEVICE NOVALED GMBH (DE) 2024-06-20 WO disclosed
WO-2024126528-A1 ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING A COMPOUND OF FORMULA (I) AND A COMPOUND OF FORMULA (II), AND DISPLAY DEVICE COMPRISING THE ORGANIC ELECTROLUMINESCENT DEVICE NOVALED GMBH (DE) 2024-06-20 WO disclosed
WO-2024046607-A1 ORGANIC ELECTROLUMINESCENT DEVICE COMPRISING A COMPOUND OF FORMULA (I) AND A COMPOUND OF FORMULA (II), AND DISPLAY DEVICE COMPRISING THE ORGANIC ELECTROLUMINESCENT DEVICE NOVALED GMBH (DE) 2024-03-07 WO disclosed
CN-117529476-A Preparation of substituted 1, 2-diamino heterocyclic derivatives and their use as medicaments 亚飞络思制药公司 2024-02-06 CN disclosed
US-11844758-B2 Therapeutically active compounds and their methods of use SERVIER PHARMACEUTICALS LLC (US) 2023-12-19 US disclosed
EP-1246802-B1 4-AMINOPICOLINATES AND THEIR USE AS HERBICIDES DOW AGROSCIENCES LLC (US) 2007-03-14 EP disclosed
CN-1281591-C 4-aminopyridinecarboxylates and their use as herbicides DOW AGROSCIENCES LLC (US) 2006-10-25 CN disclosed
EP-1498413-A1 4-Aminopicolinates and their use as herbicides Dow AgroSciences LLC (US) 2005-01-19 EP disclosed
CN-1416419-A 4-aminopyridinecarboxylates and their use as herbicides DOW AGROSCIENCES LLC (US) 2003-05-07 CN disclosed
EP-1246802-A1 4-AMINOPICOLINATES AND THEIR USE AS HERBICIDES Dow Agrosciences LLC (US) 2002-10-09 EP disclosed
US-20010047099-A1 4-aminopicolinates and their use as herbicides DOW AGROSCIENCES LLC 2001-11-29 US disclosed
US-6297197-B1 DEMONSTRATING A BROAD SPECTRUM OF WEED CONTROL. DOW AGROSCIENCES LLC 2001-10-02 US disclosed
WO-2001051468-A1 4-AMINOPICOLINATES AND THEIR USE AS HERBICIDES DOW AGROSCIENCES LLC (US) 2001-07-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12433895-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT CTSS 115/4885IRAK4 2978/4885P2RX7 3486/4885
US-11844758-B2 Therapeutically active compounds and their methods of use MCL1, TP53, BRDT CTSS 115/4885IRAK4 2978/4885P2RX7 3486/4885
US-20240335448-A1 THERAPEUTICALLY ACTIVE COMPOUNDS AND THEIR METHODS OF USE MCL1, TP53, BRDT CTSS 115/4885IRAK4 2978/4885P2RX7 3486/4885
US-20010047099-A1 4-aminopicolinates and their use as herbicides AADAT, ABAT, DDT CTSS 3363/4885IRAK4 3446/4885P2RX7 1463/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.