SCHEMBL14468359

SCHEMBL14468359

CCCCOC(=O)c1ccc2c(c1C)CC[C@@H]2NC(=O)c1cc(C(=O)NCc2ccc(F)c(F)c2)nc2cc(C(N)=O)nn12

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 9/20 0.52
ADAMTS4 O75173 2/20 0.52
MMP3 P08254 2/20 0.52
MMP8 P22894 1/20 0.48
MMP12 P39900 1/20 0.48
S1PR3 Q99500 4/20 0.34
CRBN Q96SW2 1/20 0.33
MET P08581 1/20 0.31
CHRM4 P08173 2/20 0.31
KLKB1 P03952 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14468358 0.95 MMP13 (0.53) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL14345596 0.91 MMP13 (0.57) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL5425633 0.89 MMP13 (0.55) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL10168058 0.89 MMP13 (0.64) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL14446795 0.87 MMP13 (0.54) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL10167293 0.85 MMP13 (0.64) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL10167869 0.84 MMP13 (0.66) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL5423763 0.84 MMP13 (0.56) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL10166977 0.84 MMP13 (0.59) MMP13ADAMTS4MMP3MMP8MMP12
SCHEMBL14446794 0.83 MMP13 (0.54) MMP13ADAMTS4MMP3MMP8MMP12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070155737-A1 Heterobicyclic metalloprotease inhibitors ALANTOS PHARMACEUTICALS, INC. 2007-07-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070155737-A1 Heterobicyclic metalloprotease inhibitors ADAMTS4, ADAMTS1, ADAMTS5 MMP13 38/4885ADAMTS4 1/4885MMP3 33/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.