SCHEMBL1448079

SCHEMBL1448079

COc1ccc2c(c1)[N]CC=C2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.39
CYP11B2 P19099 3/20 0.39
GAA P10253 2/20 0.36
TRPA1 O75762 1/20 0.36
HTR2C P28335 1/20 0.36
CA2 P00918 3/20 0.35
CA12 O43570 2/20 0.35
CA1 P00915 2/20 0.35
CA7 P43166 2/20 0.35
CA9 Q16790 2/20 0.35
CA14 Q9ULX7 2/20 0.35
MAOA P21397 1/20 0.35
MAOB P27338 1/20 0.35
CA5A P35218 1/20 0.35
NOS3 P29474 1/20 0.35
NOS1 P29475 1/20 0.35
NOS2 P35228 1/20 0.35
CYP19A1 P11511 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2A6 P11509 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1447451 0.86 HTR2C (0.36) CYP11B1CYP11B2GAATRPA1HTR2C
SCHEMBL322514 0.72 TRPA1 (0.39) CYP11B1CYP11B2GAATRPA1CA2
SCHEMBL4133299 0.68 GAA (0.50) CYP11B1CYP11B2GAACA2CA12
SCHEMBL31463289 0.68 GAA (0.50) CYP11B1CYP11B2GAACA2CA12
SCHEMBL28445528 0.68 STS (0.60) CYP11B1CYP11B2GAATRPA1HTR2C
SCHEMBL29634256 0.68 STS (0.60) CYP11B1CYP11B2GAATRPA1HTR2C
SCHEMBL3840318 0.68 GAA (0.40) CYP11B1CYP11B2GAATRPA1CA2
SCHEMBL1447442 0.68 CHRNB2 (0.38) HTR2CCA9NOS3NOS1NOS2
SCHEMBL28878034 0.66 KDM4E (0.42) GAACA2CA12CA1CA7
SCHEMBL1479378 0.66 MAOA (0.50) CYP11B1CYP11B2GAAMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4201923-A1 5-SUBSTITUTED 2,3-DIHYDROPYRIDIN-4-ONES AND PROCESS FOR PREPARING THE SAME Karl-Franzens-Universität Graz (AT) 2023-06-28 EP disclosed
EP-3666757-A1 PROCESS FOR PREPARING A PIPERIDIN-4-ONE Karl-Franzens-Universität Graz (AT) 2020-06-17 EP disclosed
EP-2301627-A1 Novel antimalarial 3-azabicyclo[3.2.2]nonane derivatives University of Graz (AT) 2011-03-30 EP disclosed