SCHEMBL14489202

SCHEMBL14489202

CBc1ccc([C@H]2c3cc(C#N)ccc3C[C@@H]2C)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 4/20 0.36
DRD3 P35462 3/20 0.36
PNMT P11086 6/20 0.34
HTR2A P28223 1/20 0.34
HTR2C P28335 1/20 0.34
HTR2B P41595 1/20 0.34
TRPM5 Q9NZQ8 1/20 0.33
SLC22A12 Q96S37 1/20 0.32
CHRNA1 P02708 1/20 0.32
CHRNG P07510 1/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB2 P17787 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNA4 P43681 1/20 0.32
CHRND Q07001 1/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
SLC6A3 Q01959 1/20 0.32
LRRK2 Q5S007 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14489427 0.89 PNMT (0.38) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489151 0.84 TRPM5 (0.41) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489010 0.83 DRD2 (0.38) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489506 0.82 KDM1A (0.43) HTR2AHTR2CHTR2BSLC6A4KDM1A
SCHEMBL14489381 0.82 DRD2 (0.36) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489380 0.80 DRD2 (0.40) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14488879 0.78 SLC6A4 (0.39) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489288 0.76 DRD3 (0.41) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489294 0.76 HTR2C (0.36) DRD2DRD3PNMTHTR2AHTR2C
SCHEMBL14489263 0.75 TRPM5 (0.42) HTR2AHTR2CHTR2BTRPM5SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007073503-A2 INDANE MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-KB ACTIVITY AND USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-28 WO disclosed