SCHEMBL14489294

SCHEMBL14489294

Cc1cccc([C@H]2c3cc(C#N)ccc3C[C@@H]2C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.36
AR P10275 1/20 0.36
CHRNA1 P02708 1/20 0.35
CHRNG P07510 1/20 0.35
CHRNB1 P11230 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
CHRND Q07001 1/20 0.35
SIRT2 Q8IXJ6 1/20 0.34
PNMT P11086 1/20 0.34
DRD2 P14416 4/20 0.34
DRD3 P35462 3/20 0.34
HTR2A P28223 1/20 0.34
HTR2B P41595 1/20 0.34
TRPM5 Q9NZQ8 2/20 0.33
MAOB P27338 1/20 0.33
IDO1 P14902 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14489380 0.91 DRD2 (0.40) HTR2CCHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL14489288 0.87 DRD3 (0.41) HTR2CCHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL14489010 0.86 DRD2 (0.38) HTR2CCHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL14489263 0.86 TRPM5 (0.42) HTR2CHTR2AHTR2BTRPM5
SCHEMBL14489427 0.83 PNMT (0.38) HTR2CCHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL14488879 0.81 SLC6A4 (0.39) HTR2CPNMTDRD2DRD3HTR2A
SCHEMBL14489381 0.79 DRD2 (0.36) HTR2CPNMTDRD2DRD3HTR2A
SCHEMBL14489151 0.78 TRPM5 (0.41) HTR2CCHRNA1CHRNGCHRNB1CHRNB2
SCHEMBL14489506 0.76 KDM1A (0.43) HTR2CARHTR2AHTR2BMAOB
SCHEMBL14489202 0.76 DRD2 (0.36) HTR2CCHRNA1CHRNGCHRNB1CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007073503-A2 INDANE MODULATORS OF GLUCOCORTICOID RECEPTOR, AP-1, AND/OR NF-KB ACTIVITY AND USE THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2007-06-28 WO disclosed