SCHEMBL145233

SCHEMBL145233

CCCCC(CCCC)c1ccnc(-c2cc(C(CCCC)CCCC)cc(-c3cc(C(CCCC)CCCC)ccn3)n2)c1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 2/20 0.33
CCR5 P51681 2/20 0.33
CCR8 P51685 2/20 0.33
TLR8 Q9NR97 2/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
BDKRB2 P30411 2/20 0.32
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP19A1 P11511 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
IDO1 P14902 1/20 0.30
CTRC Q99895 1/20 0.30
BRS3 P32247 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL175672 0.93 CCR1 (0.38) CCR1CCR5CCR8ALDH1A1POLB
Bromide SCHEMBL2514869 0.90 CCR1 (0.35) CCR1CCR5CCR8ALDH1A1POLB
SCHEMBL174988 0.87 NR1I2 (0.39) CCR1CCR5CCR8BDKRB2
SCHEMBL3040111 0.87 NR1I2 (0.39) CCR1CCR5CCR8ALDH1A1POLB
SCHEMBL2511650 0.83 KDM5A (0.35) ALDH1A1POLBBRS3
SCHEMBL13039644 0.82 LNPEP (0.37) MAPT
SCHEMBL5974098 0.81 NR1I2 (0.47) CCR1CCR5CCR8BDKRB2
SCHEMBL6417924 0.80 KDM5A (0.50)
SCHEMBL2136994 0.78 ALDH1A1 (0.35) CCR1CCR5CCR8ALDH1A1
Bromide SCHEMBL2521169 0.78 POLB (0.35) ALDH1A1POLBMAPTCYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 203 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3042645-B2 Dental composites with improved storage stability IVOCLAR VIVADENT AG (LI) 2025-03-12 EP claimed
US-20230399450-A1 PREPARATION OF NON-POLAR-POLAR BLOCK COPOLYMERS VIA VINYL-TERMINATED POLYOLEFINS DOW GLOBAL TECHNOLOGIES LLC (US) 2023-12-14 US claimed
EP-4244263-A1 PREPARATION OF NON-POLAR-POLAR BLOCK COPOLYMERS VIA VINYL-TERMINATED POLYOLEFINS Dow Global Technologies LLC (US) 2023-09-20 EP claimed
US-11357708-B2 Dental composites with improved storage stability IVOCLAR VIVADENT AG (LI) 2022-06-14 US claimed
WO-2022103803-A1 PREPARATION OF NON-POLAR–POLAR BLOCK COPOLYMERS VIA VINYL-TERMINATED POLYOLEFINS DOW GLOBAL TECHNOLOGIES LLC (US) 2022-05-19 WO claimed
EP-3042645-B1 Dental composites with improved storage stability IVOCLAR VIVADENT AG (LI) 2022-04-27 EP claimed
US-20210309880-A1 DIRECT TO SUBSTRATE COATING VIA IN SITU POLYMERIZATION HENKEL AG & CO. KGAA (DE) 2021-10-07 US claimed
WO-2020131445-A1 DIRECT TO SUBSTRATE COATING VIA IN SITU POLYMERIZATION HENKEL AG & CO. KGAA (DE) 2020-06-25 WO claimed
US-20180318178-A1 DENTAL COMPOSITES WITH IMPROVED STORAGE STABILITY IVOCLAR VIVADENT AG (LI) 2018-11-08 US claimed
EP-3397276-A1 ANTIBODIES AND CONJUGATES THEREOF Kodiak Sciences Inc. (US) 2018-11-07 EP claimed
EP-3310847-A1 METHOD OF PREPARING A POLYROTAXANE AND POLYROTAXANE Universität des Saarlandes (DE) 2018-04-25 EP claimed
WO-2017117464-A1 ANTIBODIES AND CONJUGATES THEREOF KODIAK SCIENCES INC. (US) 2017-07-06 WO claimed
WO-2016202906-A1 METHOD OF PREPARING A POLYROTAXANE AND POLYROTAXANE UNIVERSITAET DES SAARLANDES (DE) 2016-12-22 WO claimed
EP-3042645-A1 Dental composites with improved storage stability Ivoclar Vivadent AG (LI) 2016-07-13 EP claimed
EP-2850115-A1 POLYCARBONATE COPOLYMERS VIA CONTROLLED RADICAL POLYMERIZATION SABIC Innovative Plastics IP B.V. (NL) 2015-03-25 EP claimed
US-8975346-B2 Polycarbonate copolymers via controlled radical polymerization SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2015-03-10 US claimed
US-20130310524-A1 Polycarbonate Copolymers Via Controlled Radical Polymerization SABIC GLOBAL TECHNOLOGIES B.V. (NL) 2013-11-21 US claimed
WO-2013171634-A1 POLYCARBONATE COPOLYMERS VIA CONTROLLED RADICAL POLYMERIZATION SABIC INNOVATIVE PLASTICS IP B.V. (NL) 2013-11-21 WO claimed
EP-4724108-A2 COMPOSITIONS OF CONJUGATED AND UNCONJUGATED PROTEINS Kodiak Sciences Inc. (US) 2026-04-15 EP disclosed
WO-1999050310-A1 APPLICATION OF ATOM TRANSFER RADICAL POLYMERIZATION TO WATER-BORNE POLYMERIZATION SYSTEMS CARNEGIE MELLON UNIVERSITY (US) 1999-10-07 WO disclosed