SCHEMBL14542007

SCHEMBL14542007

COc1ccc(Cn2nc(C)c(-c3ccccc3N=O)c(CCc3cccc(F)c3)c2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CASR P41180 2/20 0.38
GAA P10253 2/20 0.37
POLB P06746 1/20 0.36
AURKA O14965 1/20 0.36
AURKB Q96GD4 1/20 0.36
ALDH1A1 P00352 2/20 0.36
PKM P14618 1/20 0.36
CES2 O00748 1/20 0.36
TP53 P04637 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
THRB P10828 1/20 0.36
HPGD P15428 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5313301 0.88 CASR (0.49) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5313082 0.85 LMNA (0.45) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5307935 0.83 TP53 (0.44) MAPTCASRPOLBALDH1A1TP53
SCHEMBL5312354 0.82 TP53 (0.42) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL5307893 0.81 THRB (0.41) MAPTCASRPOLBALDH1A1TP53
SCHEMBL5315681 0.81 CASR (0.49) CASRGAAPOLBALDH1A1PKM
SCHEMBL5307948 0.81 CASR (0.49) CASRGAAPOLBAURKAAURKB
SCHEMBL5312353 0.79 CASR (0.54) CASRGAAPOLB
SCHEMBL5308342 0.79 POLB (0.48) MAPTCASRPOLBALDH1A1TP53
SCHEMBL5310910 0.79 CASR (0.52) CASRPOLBALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044796-A2 PYRIDAZINONE COMPOUNDS AS CALCILYTICS NPS PHARMACEUTICALS, INC. (US) 2007-04-19 WO disclosed