SCHEMBL14565740

SCHEMBL14565740

N#Cc1ccccc1S(=O)(=O)N1CCCC(NC=O)C(=O)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.47
PKM P14618 1/20 0.45
HTR2A P28223 1/20 0.41
HTR2C P28335 1/20 0.41
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.40
GPR183 P32249 1/20 0.39
CTDSP1 Q9GZU7 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
MAPT P10636 1/20 0.39
JAK2 O60674 1/20 0.38
JAK1 P23458 1/20 0.38
GBA1 P04062 2/20 0.37
TSHR P16473 2/20 0.37
GAA P10253 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14565738 0.83 KMT2A (0.48) HTR2AHTR2CALDH1A1L3MBTL1TSHR
SCHEMBL14565729 0.81 PKM (0.46) PKMKDM4EALDH1A1GAA
SCHEMBL14565743 0.81 MEN1 (0.55) HTR2AHTR2CMAPTTSHR
SCHEMBL5105476 0.80 ATM (0.52) ATMPKMHTR2AHTR2CKDM4E
SCHEMBL4767334 0.78 ATM (0.44) ATMPKMHTR2AHTR2CKDM4E
SCHEMBL14565734 0.76 CTSK (0.49) PKM
SCHEMBL4767042 0.75 ATM (0.42) ATMPKMHTR2AHTR2CKDM4E
SCHEMBL4898677 0.75 CTSK (0.47) ATMPKMKDM4E
SCHEMBL14565744 0.75 PKM (0.49) PKMKDM4EALDH1A1L3MBTL1TSHR
SCHEMBL1014809 0.75 PKM (0.67) ATMPKMHTR2AHTR2CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196099-B2 Compounds and compositions as cathepsin inhibitors AVENTIS PHARMACEUTICALS INC. (US) 2007-03-27 US disclosed