Maleic Acid

Maleic Acid

SCHEMBL1463346

C=Cc1ccc(S(=O)(=O)O)cc1.O=C(O)/C=C\C(=O)O

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 known ✓ P27487 2/20 0.37
TDP1 Q9NUW8 2/20 0.78
TSHR P16473 3/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
LMNA P02545 2/20 0.42
ALDH1A1 P00352 6/20 0.41
NT5E P21589 1/20 0.41
GAA P10253 2/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 2/20 0.39
CYP2D6 P10635 1/20 0.39
PKM P14618 2/20 0.37
HCAR2 Q8TDS4 2/20 0.37
CA12 O43570 2/20 0.37
AKR1B10 O60218 2/20 0.37
CA1 P00915 2/20 0.37
CA2 P00918 2/20 0.37
CA3 P07451 2/20 0.37
AKR1B1 P15121 2/20 0.37
CA4 P22748 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL1463348 1.00 TDP1 (0.78) TDP1TSHRSMN1; SMN2LMNAALDH1A1
Acrylic Acid SCHEMBL3406953 0.91 TDP1 (0.81) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL31126649 0.88 TDP1 (1.00) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL452529 0.88 TDP1 (1.00) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL25711 0.88 TDP1 (1.00) TDP1TSHRSMN1; SMN2LMNAALDH1A1
Acrylic Acid SCHEMBL28117148 0.87 TDP1 (0.75) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL331672 0.86 TDP1 (0.95) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL2121269 0.86 TDP1 (0.95) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL2198423 0.86 TDP1 (0.95) TDP1TSHRSMN1; SMN2LMNAALDH1A1
SCHEMBL17476625 0.86 TDP1 (0.95) TDP1TSHRSMN1; SMN2LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2480666-B1 COMPOSITIONS, METHODS, AND KITS FOR ISOLATING AND ANALYZING NUCLEIC ACIDS USING AN ANION EXCHANGE MATERIAL QIAGEN GAITHERSBURG INC (US) 2017-03-08 EP disclosed
US-9505713-B2 High-purity sodium p-styrenesulfonate with excellent hue, method for producing the same, poly(sodium p-styrenesulfonate) with excellent hue using the same, and dispersant and synthetic starch for clothing finishing using the poly(sodium p-styrenesulfonate) TOSOH ORGANIC CHEMICAL CO., LTD (JP) 2016-11-29 US disclosed
US-9238809-B2 Compositions, methods, and kits for isolating and analyzing nucleic acids using an anion exchange material QIAGEN GAITHERSBURG, INC. (US) 2016-01-19 US disclosed
US-20150246876-A1 HIGH-PURITY SODIUM P-STYRENESULFONATE WITH EXCELLENT HUE, METHOD FOR PRODUCING THE SAME, POLY (SODIUM P-STYRENESULFONATE) WITH EXCELLENT HUE USING THE SAME, AND DISPERSANT AND SYNTHETIC STARCH FOR CLOTHING FINISHING USING THE POLY ( SODIUM P-STYRENESULFONATE) TOSOH ORGANIC CHEMICAL CO., LTD. (JP) 2015-09-03 US disclosed
CN-102712946-A Sensor layers and methods related thereto EDWARDS LIFESCIENCES CORP 2012-10-03 CN disclosed
EP-2480666-A1 COMPOSITIONS, METHODS, AND KITS FOR ISOLATING AND ANALYZING NUCLEIC ACIDS USING AN ANION EXCHANGE MATERIAL QIAGEN Gaithersburg, Inc. (US) 2012-08-01 EP disclosed
WO-2011037692-A1 COMPOSITIONS, METHODS, AND KITS FOR ISOLATING AND ANALYZING NUCLEIC ACIDS USING AN ANION EXCHANGE MATERIAL QIAGEN GAITHERSBURG INC. (US) 2011-03-31 WO disclosed
US-20110071031-A1 COMPOSITIONS, METHODS, AND KITS FOR ISOLATING AND ANALYZING NUCLEIC ACIDS USING AN ANION EXCHANGE MATERIAL QIAGEN GAITHERSBURG INC. (US) 2011-03-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150246876-A1 HIGH-PURITY SODIUM P-STYRENESULFONATE WITH EXCELLENT HUE, METHOD FOR PRODUCING THE SAME, POLY (SODIUM P-STYRENESULFONATE) WITH EXCELLENT HUE USING THE SAME, AND DISPERSANT AND SYNTHETIC STARCH FOR CLOTHING FINISHING USING THE POLY ( SODIUM P-STYRENESULFONATE) HPSE, STS, TST DPP4 4717/4885TDP1 2501/4885TSHR 2827/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.