SCHEMBL14656256

SCHEMBL14656256

CC(=O)c1cc2c(O)c3ccccc3c(O)c2o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.50
MAPT P10636 4/20 0.50
ALDH1A1 P00352 4/20 0.50
GAA P10253 3/20 0.50
HSD17B10 Q99714 3/20 0.50
MEN1 O00255 2/20 0.50
POLB P06746 2/20 0.50
KMT2A Q03164 2/20 0.50
ALOX12 P18054 2/20 0.50
KDM4C Q9H3R0 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
NSD2 O96028 1/20 0.46
MCL1 Q07820 1/20 0.46
CA12 O43570 1/20 0.45
CA9 Q16790 1/20 0.45
LMNA P02545 2/20 0.43
RECQL P46063 1/20 0.43
STAT3 P40763 3/20 0.42
HPGD P15428 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22079874 0.82 ALDH1A1 (0.51) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL12527554 0.79 KLKB1 (0.43) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL12526833 0.79 KDM4E (0.39) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL18123592 0.78 KDM4E (0.38) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL18123831 0.78 KDM4E (0.38) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL18123699 0.77 MAPT (0.37) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL18123783 0.77 MAPT (0.37) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL28661959 0.76 ALDH1A1 (0.41) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL20851793 0.76 LMNA (0.43) KDM4EMAPTALDH1A1GAAHSD17B10
SCHEMBL15200611 0.76 ALOX15 (0.41) KDM4EMAPTALDH1A1GAAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107311969-B Novel compounds and compositions for targeting cancer stem cells 北京强新生物科技有限公司 2022-01-28 CN claimed
CN-104080449-A Method for preparing aqueous mano particle suspensions of derivatives of 4,9-dihydroxy-naphtho[2,3-b]furan aliphatic acid esters ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO LTD 2014-10-01 CN claimed
CN-107721958-B Novel compounds and compositions for targeting cancer stem cells 北京强新生物科技有限公司 2024-08-23 CN disclosed
EP-2547205-B1 NOVEL METHODS FOR TARGETING CANCER STEM CELLS 1GLOBE BIOMEDICAL CO LTD (CN) 2024-03-20 EP disclosed
CN-107375260-B Novel compounds and compositions for targeting cancer stem cells 北京强新生物科技有限公司 2023-10-24 CN disclosed
CN-107311969-B Novel compounds and compositions for targeting cancer stem cells 北京强新生物科技有限公司 2022-01-28 CN disclosed
CN-106211758-B Use of 2-acetylnaphtho [2,3-b ] furan-4, 9-dione for treating cancer 北京强新生物科技有限公司 2021-03-23 CN disclosed
US-20200397740-A1 2-ACETYLNAPHTHO[2,3-B]FURAN -4,9-DIONE FOR USE ON TREATING CANCER Sumitomo Dainnipon Pharma Oncology. Inc. (US) 2020-12-24 US disclosed
US-20200392098-A1 SUBSTITUTED NAPHTHO[2,3-b]FURANS AS WATER-SOLUBLE PRODRUGS FOR PREVENTING AND/OR TREATING CANCER BOSTON BIOMEDICAL, INC. (US) 2020-12-17 US disclosed
US-10800752-B2 Substituted naphtho[2,3-b]furans as water-soluble prodrugs for preventing and/or treating cancer BOSTON BIOMEDICAL, INC. (US) 2020-10-13 US disclosed
US-10543189-B2 2-acetylnaphtho[2,3-b]furan -4,9-dione for use on treating cancer BOSTON BIOMEDICAL, INC. (US) 2020-01-28 US disclosed
US-20150183756-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TARGETING CANCER STEM CELLS BOSTON BIOMEDICAL, INC. (US) 2015-07-02 US disclosed
US-20150164794-A1 METHOD FOR PREPARING AQUEOUS NANOPARTICLE SUSPENSIONS OF DERIVATIVES OF 4,9-DIHYDROXY-NAPHTHO[2,3-b]FURAN ALIPHATIC ACID ESTERS Zhoushan Haizhongzhou Xinsheng Pharmaceuticals, Co., Ltd. (CN) 2015-06-18 US disclosed
US-20150164794-A1 METHOD FOR PREPARING AQUEOUS NANOPARTICLE SUSPENSIONS OF DERIVATIVES OF 4,9-DIHYDROXY-NAPHTHO[2,3-b]FURAN ALIPHATIC ACID ESTERS Zhoushan Haizhongzhou Xinsheng Pharmaceuticals, Co., Ltd. (CN) 2015-06-18 US disclosed
EP-2814480-A1 METHOD FOR PREPARING AQUEOUS MANO PARTICLE SUSPENSIONS OF DERIVATIVES OF 4,9-DIHYDROXY-NAPHTHO[2,3-b]FURAN ALIPHATIC ACID ESTERS Zhoushan Haizhongzhou Xinsheng Pharmaceuticals Co., Ltd. (CN) 2014-12-24 EP disclosed
CN-104080449-A Method for preparing aqueous mano particle suspensions of derivatives of 4,9-dihydroxy-naphtho[2,3-b]furan aliphatic acid esters ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO LTD 2014-10-01 CN disclosed
WO-2013120229-A1 METHOD FOR PREPARING AQUEOUS MANO PARTICLE SUSPENSIONS OF DERIVATIVES OF 4,9-DIHYDROXY-NAPHTHO[2,3-b]FURAN ALIPHATIC ACID ESTERS ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO., LTD. (CN) 2013-08-22 WO disclosed
WO-2013120229-A1 METHOD FOR PREPARING AQUEOUS MANO PARTICLE SUSPENSIONS OF DERIVATIVES OF 4,9-DIHYDROXY-NAPHTHO[2,3-b]FURAN ALIPHATIC ACID ESTERS ZHOUSHAN HAIZHONGZHOU XINSHENG PHARMACEUTICALS CO., LTD. (CN) 2013-08-22 WO disclosed
US-20130034591-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TARGETING CANCER STEM CELLS BOSTON BIOMEDICAL, INC. (US) 2013-02-07 US disclosed
US-20130028944-A1 NOVEL METHODS FOR TARGETING CANCER STEM CELLS BOSTON BIOMEDICAL, INC. (US) 2013-01-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130034591-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TARGETING CANCER STEM CELLS MCL1, DDX21, TP53 KDM4E 4028/4885MAPT 2203/4885ALDH1A1 259/4885
US-20130028944-A1 NOVEL METHODS FOR TARGETING CANCER STEM CELLS DDX21, MCL1, SNX2 KDM4E 4089/4885MAPT 2925/4885ALDH1A1 173/4885
US-20200392098-A1 SUBSTITUTED NAPHTHO[2,3-b]FURANS AS WATER-SOLUBLE PRODRUGS FOR PREVENTING AND/OR TREATING CANCER NR0B1, NR0B2, NR2C2 KDM4E 3479/4885MAPT 4840/4885ALDH1A1 716/4885
US-20150164794-A1 METHOD FOR PREPARING AQUEOUS NANOPARTICLE SUSPENSIONS OF DERIVATIVES OF 4,9-DIHYDROXY-NAPHTHO[2,3-b]FURAN ALIPHATIC ACID ESTERS FASN, NCDN, NCL KDM4E 3672/4885MAPT 1903/4885ALDH1A1 114/4885
US-20200397740-A1 2-ACETYLNAPHTHO[2,3-B]FURAN -4,9-DIONE FOR USE ON TREATING CANCER B3GNT2, NAT1, NQO1 KDM4E 3905/4885MAPT 2559/4885ALDH1A1 65/4885
US-10800752-B2 Substituted naphtho[2,3-b]furans as water-soluble prodrugs for preventing and/or treating cancer NR0B1, NR0B2, NR2C2 KDM4E 3479/4885MAPT 4840/4885ALDH1A1 716/4885
US-20150183756-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR TARGETING CANCER STEM CELLS MCL1, DDX21, TP53 KDM4E 4028/4885MAPT 2203/4885ALDH1A1 259/4885
US-10543189-B2 2-acetylnaphtho[2,3-b]furan -4,9-dione for use on treating cancer B3GNT2, NAT1, NQO1 KDM4E 3905/4885MAPT 2559/4885ALDH1A1 65/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.