SCHEMBL14720472

SCHEMBL14720472

CCOCCS(=O)(=O)c1ccc(C=C2CCN(C3CCC3)CC2)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.38
POLB P06746 1/20 0.38
LOX P28300 1/20 0.37
TP53 P04637 1/20 0.36
MLNR O43193 1/20 0.35
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
KCNH2 Q12809 1/20 0.34
HRH3 Q9Y5N1 5/20 0.34
KDM2B Q8NHM5 2/20 0.34
CYP2D6 P10635 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14720768 0.89 KCNH2 (0.44) ALDH1A1POLBLOXTP53MLNR
SCHEMBL14720573 0.85 SRD5A2 (0.37) ALDH1A1POLBMLNRHRH3CYP2D6
SCHEMBL14720491 0.85 HRH3 (0.45) ALDH1A1POLBTP53MLNRKDM4E
SCHEMBL14721060 0.76 KCNH2 (0.43) ALDH1A1TP53KDM4EKCNH2HRH3
SCHEMBL14720551 0.73 ALDH1A1 (0.56) ALDH1A1POLBNPC1
SCHEMBL14720578 0.72 KDM4E (0.47) ALDH1A1POLBKDM4EGAAHRH3
SCHEMBL14720718 0.72 HSD11B1 (0.51) ALDH1A1POLBKDM4EGAAKCNH2
SCHEMBL14720724 0.70 ALDH1A1 (0.58) ALDH1A1POLBKMT2ANPC1
SCHEMBL14720887 0.70 POLB (0.52) ALDH1A1POLBKDM4EGAAMEN1
SCHEMBL14720486 0.70 NAMPT (0.38) ALDH1A1KDM4EHRH3KDM2BMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO claimed
WO-2013027001-A1 COMPOUNDS AND THEIR USE TO TREAT HISTAMINE H3 RELATED DISORDERS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-02-28 WO disclosed