SCHEMBL14722260

SCHEMBL14722260

COc1ccc(C2=CC(=O)COc3c2cc(OC)c(OC)c3OC)cc1NC(=O)OC(C)(C)C

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 3/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
TSHR P16473 2/20 0.33
MAPT P10636 3/20 0.33
CTSL P07711 2/20 0.33
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
LMNA P02545 1/20 0.33
TUBB4A P04350 1/20 0.33
TUBB P07437 1/20 0.33
TUBA3C P0DPH7 1/20 0.33
TUBA1B P68363 1/20 0.33
TUBA4A P68366 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721668 0.88 MAPT (0.37) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL14722027 0.87 TSHR (0.43) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL14722029 0.85 PDE3B (0.35) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL14725529 0.84 MMP1 (0.35) ALDH1A1KDM4ESMN1; SMN2MAPTCTSL
SCHEMBL14725391 0.83 SMN1; SMN2 (0.35) ALDH1A1KDM4ESMN1; SMN2RAB9ATSHR
SCHEMBL14722118 0.82 ALDH1A1 (0.35) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL14725496 0.82 ALDH1A1 (0.33) ALDH1A1KDM4ESMN1; SMN2NPC1RAB9A
SCHEMBL14721811 0.79 TUBB4A (0.48) ALDH1A1KDM4ETDP1MAPTTP53
SCHEMBL14723189 0.79 TUBB4A (0.43) TUBB4ATUBBTUBA3CTUBA1BTUBA4A
Hydrochloric Acid SCHEMBL14722160 0.78 TUBB4A (0.43) ALDH1A1MAPTMEN1KMT2ATUBB4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed