SCHEMBL14725529

SCHEMBL14725529

COc1ccc(C2=CC(=O)CCc3c2cc(OC)c(OC)c3OC)cc1NC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.35
MMP2 P08253 1/20 0.35
MMP9 P14780 1/20 0.35
MMP8 P22894 1/20 0.35
MMP13 P45452 1/20 0.35
ALDH1A1 P00352 2/20 0.34
GAA P10253 1/20 0.34
CTSL P07711 1/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
PIK3CD O00329 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
KDR P35968 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CG P48736 1/20 0.33
BACE1 P56817 1/20 0.33
PRKDC P78527 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14721210 0.87 KDM4E (0.37) ALDH1A1KDM4EHPGDMEN1KMT2A
SCHEMBL14725517 0.86 AAK1 (0.44) ALDH1A1CTSLMEN1KMT2AMAPT
SCHEMBL14725525 0.84 BTK (0.37) ALDH1A1GAAPIK3CDABL1EGFR
SCHEMBL14722260 0.84 ALDH1A1 (0.34) ALDH1A1GAACTSLKDM4EMEN1
SCHEMBL14721722 0.84 TSHR (0.36) MMP1MMP2MMP9MMP8MMP13
SCHEMBL14721726 0.84 TSHR (0.36) MMP1MMP2MMP9MMP8MMP13
SCHEMBL14721721 0.81 NPSR1 (0.30)
SCHEMBL14725450 0.79 AAK1 (0.43)
SCHEMBL14721685 0.79 AAK1 (0.43)
SCHEMBL14725511 0.78 SRC (0.40) ALDH1A1GAACTSLKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed