SCHEMBL14725517

SCHEMBL14725517

COc1ccc(C2=CC(=O)CCc3c2cc(OC)c(OC)c3OC)cc1NC(=O)C(CC(C)C)NC(=O)OC(C)(C)C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 4/20 0.44
TSHR P16473 1/20 0.42
MAP1LC3B Q9GZQ8 1/20 0.39
MAP1LC3A Q9H492 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 1/20 0.36
MAPT P10636 1/20 0.36
RAB9A P51151 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
ANPEP P15144 1/20 0.35
SRC P12931 1/20 0.35
CTSL P07711 2/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14725511 0.88 SRC (0.40) AAK1TSHRMAP1LC3BMAP1LC3AMEN1
SCHEMBL14725528 0.88 REN (0.40) REN
SCHEMBL14722027 0.87 TSHR (0.43) AAK1TSHRMAP1LC3BMAP1LC3AMEN1
SCHEMBL14725529 0.86 MMP1 (0.35) MEN1KMT2ASMN1; SMN2ALDH1A1MAPT
SCHEMBL14725450 0.84 AAK1 (0.43) AAK1TSHR
SCHEMBL14721685 0.84 AAK1 (0.43) AAK1TSHR
SCHEMBL14725433 0.81 TSHR (0.38) AAK1TSHRMEN1KMT2ASMN1; SMN2
SCHEMBL14725494 0.79 PSEN1 (0.42) REN
SCHEMBL14721210 0.78 KDM4E (0.37) TSHRMEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL14725251 0.76 S1PR1 (0.35) MEN1KMT2ASMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013026942-A1 TUBULIN BINDING AGENTS THE PROVOST, FELLOWS, FOUNDATION SCHOLARS, AND THE OTHER MEMBERS OF BOARD, OF THE COLLEGE OF THE HOLY AND UNDIVIDED TRINITY OF QUEEN ELIZABETH, NEAR DUBLIN (IE) 2013-02-28 WO disclosed