SCHEMBL14732158

SCHEMBL14732158

CCc1c(Br)cccc1C=C1CCN(CC(=O)O)CC1

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
OGA O60502 3/20 0.33
MCHR1 Q99705 3/20 0.33
EP300 Q09472 2/20 0.32
CARM1 Q86X55 2/20 0.32
S1PR1 P21453 1/20 0.32
ALDH1A1 P00352 2/20 0.32
GLA P06280 1/20 0.32
S1PR3 Q99500 1/20 0.32
S1PR5 Q9H228 1/20 0.32
NLRP3 Q96P20 1/20 0.32
KDM4E B2RXH2 1/20 0.31
SLC6A9 P48067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2591378 0.86 KMT2A (0.41) MEN1KMT2AS1PR1ALDH1A1KDM4E
SCHEMBL1293181 0.80 SRD5A2 (0.32) EP300CARM1
SCHEMBL1293824 0.80 SIGMAR1 (0.37) MEN1KMT2AALDH1A1KDM4E
SCHEMBL14732194 0.78 S1PR5 (0.34) OGAS1PR1S1PR3S1PR5
SCHEMBL1293336 0.78 GRM5 (0.45) ALDH1A1KDM4E
SCHEMBL2587701 0.75 GRM5 (0.39) MEN1KMT2AALDH1A1KDM4E
SCHEMBL1293136 0.73 PNMT (0.34)
SCHEMBL2591372 0.71
SCHEMBL1293137 0.66 LMNA (0.41) MEN1KMT2AALDH1A1
SCHEMBL16956377 0.66 GABRA1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563785-A1 COMPOUNDS AS AGONISTS OF S1P1 RECEPTORS Glaxo Group Limited (GB) 2013-03-06 EP disclosed
US-8389508-B2 Heterocyclic compounds GLAXO GROUP LIMITED (GB) 2013-03-05 US disclosed