SCHEMBL14734344

SCHEMBL14734344

COC(=O)C(C)Nc1ccc(OC)cc1[N+](=O)[O-]

nearest known ligand 0.70

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.56
RAB9A P51151 2/20 0.56
MAPK1 P28482 2/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
NPC1 O15118 1/20 0.56
AKR1C3 P42330 2/20 0.55
AKR1C2 P52895 2/20 0.55
ALDH1A1 P00352 1/20 0.55
THRB P10828 1/20 0.55
LMNA P02545 3/20 0.55
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
KCNMA1 Q12791 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5945876 0.85 CRHBP (0.58) MAPTMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL1596478 0.85 CRHBP (0.58) MAPTMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL8742125 0.85 CRHBP (0.58) MAPTMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL3322365 0.85 MAPT (0.56) MAPTRAB9AMAPK1SMN1; SMN2NPC1
SCHEMBL7362765 0.84 HCAR3 (0.58) MAPTRAB9AMAPK1SMN1; SMN2NPC1
SCHEMBL31424672 0.83 KMT2A (0.71) MAPTRAB9ANPC1ALDH1A1LMNA
SCHEMBL31607362 0.82 KMT2A (0.51) MAPTMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL31607343 0.82 KMT2A (0.51) MAPTMAPK1SMN1; SMN2ALDH1A1LMNA
SCHEMBL24202566 0.80 ALDH1A1 (0.57) MAPTRAB9AMAPK1SMN1; SMN2NPC1
SCHEMBL24202568 0.80 ALDH1A1 (0.57) MAPTRAB9AMAPK1SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013034755-A1 TRIAZOLOPYRAZINE DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS H. LUNDBECK A/S (DK) 2013-03-14 WO disclosed
WO-2013027794-A1 NOVEL COMPOUND AND USE THEREOF AS PDE10 INHIBITOR 田辺三菱製薬株式会社 (JP) 2013-02-28 WO disclosed