SCHEMBL147397

SCHEMBL147397

CC(C)(C)[Si](OCc1cc(Br)ccc1Cl)(c1ccccc1)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PTGER1 P34995 1/20 0.35
CCR5 P51681 3/20 0.34
SLC6A4 P31645 2/20 0.34
HTR6 P50406 1/20 0.34
ALDH1A1 P00352 2/20 0.34
RAB9A P51151 1/20 0.34
HTR2A P28223 1/20 0.33
KCNH2 Q12809 1/20 0.33
HTT P42858 1/20 0.32
GAA P10253 1/20 0.32
SLC16A3 O15427 1/20 0.32
SLC16A1 P53985 1/20 0.32
MCTS1 Q9ULC4 1/20 0.32
HPGD P15428 1/20 0.32
PTGFR P43088 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5672566 0.89 PYCR1 (0.35) LMNASMN1; SMN2NPSR1PTGER1CCR5
SCHEMBL6298659 0.88 PYCR1 (0.35) LMNASMN1; SMN2NPSR1PTGER1CCR5
SCHEMBL17159412 0.85 LMNA (0.37) LMNASMN1; SMN2PTGER1CCR5HTR6
SCHEMBL7015152 0.84 SYK (0.37) SMN1; SMN2SLC6A4ALDH1A1HTR2AHTT
SCHEMBL30516569 0.82 KDM5A (0.36) LMNASMN1; SMN2PTGER1CCR5ALDH1A1
SCHEMBL6132650 0.82 KDM5A (0.36) LMNASMN1; SMN2PTGER1CCR5ALDH1A1
SCHEMBL7013760 0.80 MRGPRX4 (0.34) LMNAHTTSLC16A3SLC16A1MCTS1
SCHEMBL14126456 0.80 NQO2 (0.35) LMNASMN1; SMN2PTGER1ALDH1A1GAA
SCHEMBL31533391 0.79 ABL1 (0.42) LMNAPTGER1CCR5ALDH1A1HTT
SCHEMBL195484 0.79 SLC6A4 (0.36) LMNASMN1; SMN2NPSR1PTGER1CCR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20180282363-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2018-10-04 US disclosed
US-20160108078-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2016-04-21 US disclosed
US-20160108078-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2016-04-21 US disclosed
US-20140296506-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2014-10-02 US disclosed
US-20140296506-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2014-10-02 US disclosed
US-8785403-B2 Glucopyranoside compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2014-07-22 US disclosed
US-8785403-B2 Glucopyranoside compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2014-07-22 US disclosed
US-8575114-B2 SGLT-2 inhibitors, methods of making them, and uses thereof ALBANY MOLECULAR RESEARCH, INC. (US) 2013-11-05 US disclosed
US-8575114-B2 SGLT-2 inhibitors, methods of making them, and uses thereof ALBANY MOLECULAR RESEARCH, INC. (US) 2013-11-05 US disclosed
US-20120258913-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-10-11 US disclosed
US-8202984-B2 Glucopyranoside compound MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-06-19 US disclosed
US-20120058941-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-03-08 US disclosed
US-20120058941-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2012-03-08 US disclosed
US-20110237527-A1 SGLT-2 INHIBITORS, METHODS OF MAKING THEM, AND USES THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2011-09-29 US disclosed
US-20110237527-A1 SGLT-2 INHIBITORS, METHODS OF MAKING THEM, AND USES THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2011-09-29 US disclosed
US-7943788-B2 Including the antidiabetic, antiobesity sodium glucose transport inhibitor Canagliflozin (1-( beta -D-glucopyranosyl)-4-methyl-3-[5-(4-fluorophenyl)-2-thienylmethyl]benzene) MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-05-17 US disclosed
US-7943788-B2 Including the antidiabetic, antiobesity sodium glucose transport inhibitor Canagliflozin (1-( beta -D-glucopyranosyl)-4-methyl-3-[5-(4-fluorophenyl)-2-thienylmethyl]benzene) MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-05-17 US disclosed
US-20110105424-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-05-05 US disclosed
US-20110105424-A1 GLUCOPYRANOSIDE COMPOUND MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-05-05 US disclosed
US-20050233988-A1 Novel compounds TANABE SEIYAKU CO., LTD. (JP) 2005-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120058941-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 LMNA 1887/4885SMN1; SMN2 3474/4885NPSR1 3024/4885
US-20050233988-A1 Novel compounds CYP1B1, CYP4B1, CYP2B6 LMNA 1753/4885SMN1; SMN2 3266/4885NPSR1 768/4885
US-20110237527-A1 SGLT-2 INHIBITORS, METHODS OF MAKING THEM, AND USES THEREOF SLC5A2, SLC5A1, SLC10A1 LMNA 2114/4885SMN1; SMN2 2406/4885NPSR1 3722/4885
US-20110105424-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 LMNA 1887/4885SMN1; SMN2 3474/4885NPSR1 3024/4885
US-20120258913-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 LMNA 1887/4885SMN1; SMN2 3474/4885NPSR1 3024/4885
US-20180282363-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 LMNA 1887/4885SMN1; SMN2 3474/4885NPSR1 3024/4885
US-20160108078-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 LMNA 1887/4885SMN1; SMN2 3474/4885NPSR1 3024/4885
US-20140296506-A1 GLUCOPYRANOSIDE COMPOUND UGGT1, B3GAT3, FUT6 LMNA 1887/4885SMN1; SMN2 3474/4885NPSR1 3024/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.