SCHEMBL14743642

SCHEMBL14743642

CN(CC(=O)NCc1cnccn1)c1cc(C(=O)O)cc2cc(Cl)cc(Cl)c12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.37
TDP1 Q9NUW8 1/20 0.35
CHRM4 P08173 1/20 0.35
NTRK1 P04629 1/20 0.35
VNN1 O95497 1/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP2C9 P11712 1/20 0.33
NAMPT P43490 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
TSHR P16473 1/20 0.33
HPGD P15428 1/20 0.33
ALOX15 P16050 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ITK Q08881 1/20 0.33
PIK3CA P42336 1/20 0.33
IDO1 P14902 1/20 0.33
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14743807 0.91 HPGDS (0.40) HPGDSTDP1CHRM4NTRK1GAA
SCHEMBL14743626 0.88 GAA (0.48) GAAALDH1A1TSHRHPGDALOX15
SCHEMBL14743819 0.85 LMNA (0.34) TDP1CHRM4GAAALDH1A1TSHR
SCHEMBL14743424 0.85 TDP1 (0.52) TDP1ALDH1A1CYP2C9HPGDSMN1; SMN2
SCHEMBL14743068 0.84 PSMD14 (0.38) CHRM4NTRK1ALDH1A1
SCHEMBL14743576 0.84 KMT2A (0.48) TDP1GAAALDH1A1CYP2C9HPGD
SCHEMBL14743033 0.84 TDP1 (0.41) HPGDSTDP1ALDH1A1SMN1; SMN2HTT
SCHEMBL14742993 0.83 GAA (0.34) TDP1NTRK1VNN1GAAALDH1A1
SCHEMBL14743644 0.82 TDP1 (0.40) TDP1CHRM4ALDH1A1OPRM1OPRL1
SCHEMBL14743411 0.76 TDP1 (0.50) TDP1GAAALDH1A1CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013030358-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2013-03-07 WO claimed
WO-2013030358-A1 GLYCINE B ANTAGONISTS MERZ PHARMA GMBH & CO. KGAA (DE) 2013-03-07 WO disclosed