SCHEMBL14744204

SCHEMBL14744204

Nc1cc(F)c(-c2ccccc2)c(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP2 P11137 3/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39
CYP3A4 P08684 5/20 0.38
ALDH1A1 P00352 4/20 0.38
TDP1 Q9NUW8 3/20 0.38
GAA P10253 1/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
MAOA P21397 1/20 0.38
TAAR1 Q96RJ0 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TSHR P16473 1/20 0.35
THRB P10828 1/20 0.35
TP53 P04637 1/20 0.34
CYP2A6 P11509 1/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 2/20 0.34
GLA P06280 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14746573 0.86 CYP3A4 (0.46) CYP3A4ALDH1A1TDP1GAAALOX15
SCHEMBL26633297 0.86 MAOA (0.44) MAP2ADORA2AADORA1CYP3A4ALDH1A1
SCHEMBL20108664 0.78 GABRP (0.41) CYP3A4ALDH1A1TSHRKDM4EHPGD
SCHEMBL28007815 0.77 HTT (0.47) ADORA2AADORA1CYP3A4ALDH1A1TDP1
SCHEMBL17402907 0.77 CYP3A4 (0.45) ADORA2AADORA1CYP3A4ALDH1A1TDP1
SCHEMBL16014764 0.75 PTGS2 (0.55)
SCHEMBL8974389 0.74 MAP2 (0.50) MAP2GAAHTTTSHRKDM4E
SCHEMBL16013714 0.74 CYP3A4 (0.39) ADORA2AADORA1CYP3A4ALDH1A1TDP1
SCHEMBL14747016 0.74 THRB (0.44) CYP3A4ALDH1A1TDP1GAAALOX15
SCHEMBL14744163 0.74 CYP3A4 (0.42) CYP3A4ALDH1A1HTTTAAR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013029338-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-03-07 WO disclosed